EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
2.7.11.10 | 0.000011 |
- |
7-[3-(aminomethyl)phenyl]-N,1-dimethyl-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridin-4-amine |
- |
702567 |
2.7.11.10 | 0.000011 |
- |
N,8-dimethyl-2-phenyl-8H-imidazo[4,5-d][1,3]oxazolo[5,4-b]pyridin-5-amine |
- |
702567 |
2.7.11.10 | 0.000012 |
- |
3-methoxy-N-[3-[1-methyl-4-(methylamino)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridin-7-yl]benzyl]propanamide |
- |
702567 |
2.7.11.10 | 0.000014 |
- |
N-[3-[1-methyl-4-(methylamino)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridin-7-yl]benzyl]acetamide |
- |
702567 |
2.7.11.10 | 0.000015 |
- |
4-methyl-7-methylamino-2-ethylamido-4H-imidazo[4,5-d]thiazolo[5,4-b]pyridine |
IKK-2 |
705026 |
2.7.11.10 | 0.000015 |
- |
4-methyl-7-methylamino-2-methylamido-4H-imidazo[4,5-d]thiazolo[5,4-b]pyridine |
IKK-2 |
705026 |
2.7.11.10 | 0.000015 |
- |
4-methyl-7-methylamino-2-thienylamido-4H-imidazo[4,5-d]thiazolo[5,4-b]pyridine |
IKK-2 |
705026 |
2.7.11.10 | 0.000016 |
- |
N-[[3-[8-methyl-5-(methylamino)-8H-imidazo[4,5-d]-thiazolo[5,4-b]pyridine-2-yl]phenyl]methyl]-1,2,3-thiadiazole-5-amide |
IKK-2 |
705026 |
2.7.11.10 | 0.000019 |
- |
N-(8-methyl-2-phenylimidazo[1,2-a]thieno[3,2-e]pyrazin-5-yl)ethane-1,2-diamine |
IKK-2 |
705026 |
2.7.11.10 | 0.000022 |
- |
N-[3-[1-methyl-4-(methylamino)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridin-7-yl]benzyl]butanediamide |
- |
702567 |