EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
2.6.1.16 | 0.12 |
- |
N3-(4-Methoxyfumaroyl)-L-2,3-diaminopropanoic acid |
recombinant enzyme, in 10 mM KCl, 1 mg/ml bovine serum albumin, 20 mM imidazole buffer (pH 6.8), 1 mM EDTA, 1 mM dithiothreitol, and 10% (v/v) glycerol |
706608 |
2.6.1.16 | 0.127 |
- |
methyl (2E)-4-([(2S)-2-amino-3-(methylamino)-3-oxopropyl]amino)-4-oxobut-2-enoate |
pH 7.0, 37°C |
738162 |
2.6.1.16 | 0.16 |
- |
uridine 5'-diphospho-N-acetylglucosamine |
recombinant enzyme, in 10 mM KCl, 1 mg/ml bovine serum albumin, 20 mM imidazole buffer (pH 6.8), 1 mM EDTA, 1 mM dithiothreitol, and 10% (v/v) glycerol |
706608 |
2.6.1.16 | 0.27 |
- |
(2S)-2-amino-3-([(2E)-4-oxo-4-phenylbut-2-enoyl]amino)propanoic acid |
pH 7.0, 37°C |
722052 |
2.6.1.16 | 0.45 |
- |
UDP-N-acetylglucosamine |
crude enzyme preparation, pH not specified in the publication, temperature not specified in the publication |
739575 |
2.6.1.16 | 0.52 |
- |
UDP-N-acetyl-alpha-D-glucosamine |
pH 7.0, 37°C |
722052 |
2.6.1.16 | 0.66 |
- |
(2S)-2-amino-3-(([(2R,3R)-3-benzoyloxiran-2-yl]carbonyl)amino)propanoic acid |
pH 7.0, 37°C |
722052 |
2.6.1.16 | 1.55 |
- |
uridine 5'-diphospho-N-acetyl-D-glucosamine |
wild-type, pH 6.8, 37°C |
723015 |
2.6.1.16 | 1.7 |
- |
uridine 5'-diphospho-N-acetyl-D-glucosamine |
mutant Gfa1-His6DELTA343-348, pH 6.8, 37°C |
723015 |
2.6.1.16 | 1.85 |
- |
uridine 5'-diphospho-N-acetyl-D-glucosamine |
mutant Gfa1-His6DELTA655-660, pH 6.8, 37°C |
723015 |