EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.8.1.7 | 0.0017 |
- |
4-hydroxybenzoyl-CoA |
mutant R257K, pH 7.5, 25°C |
654589 |
3.8.1.7 | 0.0024 |
- |
4-hydroxybenzoyl-CoA |
mutant R24K, pH 7.5, 25°C |
654589 |
3.8.1.7 | 0.0025 |
- |
4-hydroxybenzoyl-CoA |
wild-type enzyme, pH 7.5, 25°C |
654589 |
3.8.1.7 | 0.0031 |
- |
4-methylbenzoyl-CoA |
mutant R257K, pH 7.5, 25°C |
654589 |
3.8.1.7 | 0.0042 |
- |
4-methylbenzoyl-CoA |
wild-type enzyme, pH 7.5, 25°C |
654589 |
3.8.1.7 | 0.0062 |
- |
4-hydroxybenzoyl-CoA |
mutant R67K, pH 7.5, 25°C |
654589 |
3.8.1.7 | 0.011 |
- |
4-methylbenzoyl-CoA |
mutant R24K, pH 7.5, 25°C |
654589 |
3.8.1.7 | 0.0165 |
- |
4-hydroxybenzoyl-CoA |
mutant R24L, pH 7.5, 25°C |
654589 |
3.8.1.7 | 0.019 |
- |
4-hydroxybenzoyl-CoA |
mutant R257L, pH 7.5, 25°C |
654589 |
3.8.1.7 | 0.022 |
- |
4-methylbenzoyl-3'-dephospho-CoA |
wild-type enzyme, pH 7.5, 25°C |
654589 |