EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.5.1.135 | 0.0003 |
- |
N4-acetylcytidine |
mutant enzyme E74A, at pH 8.0 and 22°C |
758354 |
3.5.1.135 | 0.00085 |
- |
N4-benzoyl-2'-deoxycytidine |
recombinant C-terminally His6-tagged enzyme, at pH 8.0 and 22°C |
758354 |
3.5.1.135 | 0.077 |
- |
N4-acetylcytidine |
recombinant enzyme, at pH 8.0 and 22°C |
758354 |
3.5.1.135 | 0.13 |
- |
N4-acetylcytidine |
recombinant C-terminally His6-tagged enzyme, at pH 8.0 and 22°C |
758354 |
3.5.1.135 | 0.13 |
- |
N4-acetylcytidine |
recombinant N-terminally His6-tagged enzyme, at pH 8.0 and 22°C |
758354 |
3.5.1.135 | 0.15 |
- |
N4-benzoylcytidine |
recombinant C-terminally His6-tagged enzyme, at pH 8.0 and 22°C |
758354 |
3.5.1.135 | 0.2 |
- |
N4-acetylcytidine |
mutant enzyme H70A, at pH 8.0 and 22°C |
758354 |
3.5.1.135 | 0.4 |
- |
N4-acetylcytidine |
mutant enzyme D27A, at pH 8.0 and 22°C |
758354 |
3.5.1.135 | 0.7 |
- |
N4-acetylcytosine |
mutant enzyme Y89A, at pH 8.0 and 22°C |
758354 |
3.5.1.135 | 0.7 |
- |
N4-acetylcytosine |
recombinant C-terminally His6-tagged enzyme, at pH 8.0 and 22°C |
758354 |