EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.4.23.B5 | 0.00000014 |
- |
DMP323 |
pH 5.6, 37°C, recombinant enzyme |
669690 |
3.4.23.B5 | 0.0000002 |
- |
amprenavir |
substrate RSLLYPALTP, pH 5.6, 37°C |
717598 |
3.4.23.B5 | 0.00000021 |
- |
indinavir |
pH 5.6, 37°C, recombinant enzyme |
669690 |
3.4.23.B5 | 0.00000041 |
- |
ritonavir |
pH 5.6, 37°C, recombinant enzyme |
669690 |
3.4.23.B5 | 0.0000018 |
- |
atazanavir |
substrate RSLLYPALTP, pH 5.6, 37°C |
717598 |
3.4.23.B5 | 0.0000019 |
- |
KH-164 |
pH 5.6, 37°C, recombinant enzyme |
669690 |
3.4.23.B5 | 0.000002 |
- |
nelfinavir |
pH 5.6, 37°C, recombinant enzyme |
669690 |
3.4.23.B5 | 0.00001 |
- |
amprenavir |
substrate KARVnLNphEAnLG, pH 5.6, 25°C |
717598 |
3.4.23.B5 | 0.000022 |
- |
atazanavir |
substrate KARVnLNphEAnLG, pH 5.6, 25°C |
717598 |
3.4.23.B5 | 0.000028 |
- |
saquinavir |
pH 5.6, 37°C, recombinant enzyme |
669690 |