EC Number   |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
|---|
   3.4.21.B28 | 0.0000018 |
- |
acetyl-Arg-(8-amino-3,6-dioxaoctanoic acid)-Gly-L-boroPro |
in 25 mM sodium phosphate buffer, pH 7.5, containing 1.0 mM EDTA and 2% (v/v) methanol, at 22°C |
718048 |
| 3.4.21.B28 | 0.0000027 |
- |
acetyl-Arg-(8-amino-3,6-dioxaoctanoic acid)-Ser-Gly-L-boroPro |
in 25 mM sodium phosphate buffer, pH 7.5, containing 1.0 mM EDTA and 2% (v/v) methanol, at 22°C |
718048 |
| 3.4.21.B28 | 0.0000057 |
- |
acetyl-Arg-(8-amino-3,6-dioxaoctanoic acid)-D-Ala-L-boroPro |
in 25 mM sodium phosphate buffer, pH 7.5, containing 1.0 mM EDTA and 2% (v/v) methanol, at 22°C |
718048 |
| 3.4.21.B28 | 0.0000075 |
- |
[(2R)-1-[(1-oxo-1,3-dihydro-2H-isoindol-2-yl)acetyl]pyrrolidin-2-yl]-9-boronic acid |
in 50 mM Tris-HCl, 100 mM NaCl, pH 7.4, at 23°C |
678648 |
| 3.4.21.B28 | 0.000012 |
- |
[(2R)-1-[N-[(2,6-dichlorophenyl)carbonyl]glycyl]-9-pyrrolidin-2-yl]boronic acid |
in 50 mM Tris-HCl, 100 mM NaCl, pH 7.4, at 23°C |
678648 |
| 3.4.21.B28 | 0.000014 |
- |
[(2R)-1-[N-(cyclohexylcarbonyl)glycyl]pyrrolidin-2-yl]-9-boronic acid |
in 50 mM Tris-HCl, 100 mM NaCl, pH 7.4, at 23°C |
678648 |
| 3.4.21.B28 | 0.0000172 |
- |
acetyl-Arg-Gly-Gly-L-boroPro |
in 25 mM sodium phosphate buffer, pH 7.5, containing 1.0 mM EDTA and 2% (v/v) methanol, at 22°C |
718048 |
| 3.4.21.B28 | 0.00002 |
- |
[(2R)-1-[N-(cyclopentylcarbonyl)glycyl]pyrrolidin-2-yl]-9-boronic acid |
in 50 mM Tris-HCl, 100 mM NaCl, pH 7.4, at 23°C |
678648 |
| 3.4.21.B28 | 0.0000207 |
- |
acetyl-Gly-L-boroPro |
in 25 mM sodium phosphate buffer, pH 7.5, containing 1.0 mM EDTA and 2% (v/v) methanol, at 22°C |
718048 |
| 3.4.21.B28 | 0.000023 |
- |
acetyl-Gly-Pro-boronic acid |
- |
680739 |
