EC Number   |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
|---|
   3.4.21.73 | -999 |
- |
more |
inhibition kinetics |
683130 |
| 3.4.21.73 | -999 |
- |
more |
inhibition kinetics of mupain variants, overview |
731932 |
| 3.4.21.73 | -999 |
- |
more |
kinetic effects of dipeptides on the inhibition of single-chain uPA and two-chain uPA, overview. Stopped-flow kinetics of P9-NBD-labeled PAI-1, 25°C, overview |
707518 |
| 3.4.21.73 | 0.0000006 |
- |
N-[4-(aminomethyl)phenyl]-6-carbamimidoyl-4-(pyrimidin-2-ylamino)naphthalene-2-carboxamide |
pH 7.4, 37°C |
732356 |
| 3.4.21.73 | 0.000002 |
- |
phenethylsulfonamidino-D-seryl-L-alanyl(P2)-L-argininal |
pH 7.4, 37°C, compound uPA-I5 |
652910 |
| 3.4.21.73 | 0.000003 |
- |
phenethylsulfonamidino-D-seryl-L-alanyl(P2)-L-argininal |
pH 7.4, 37°C, compound uPA-I6 |
652910 |
| 3.4.21.73 | 0.000006 |
- |
phenethylsulfonamidino-D-seryl-L-alanyl(P2)-L-argininal |
pH 7.4, 37°C, compound uPA-I3 |
652910 |
| 3.4.21.73 | 0.0000077 |
- |
N-(benzylsulfonyl)-D-seryl-N-(4-carbamimidoylbenzyl)-L-alaninamide |
pH 8.8, 37°C |
731467 |
| 3.4.21.73 | 0.000009 |
- |
3-(4-chloro-1-((diaminomethylene)amino)isoquinolin-7-yl)-5-methoxybenzoic acid |
- |
667943 |
| 3.4.21.73 | 0.00001 |
- |
2-[3-(7-benzamido-4-chloro-1-oxo-1H-isochromen-3-yloxy]propyl)isothiourea hydrobromide |
pH 8.8, 25°C |
683304 |
