EC Number   |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
|---|
   3.4.21.42 | -999 |
- |
more |
first order rate inhibition kinetics |
683891 |
| 3.4.21.42 | 0.000012 |
- |
N-(3'-[[5-carbamimidoyl-2-(methylsulfanyl)thiophen-3-yl]sulfonyl]-6-methylbiphenyl-2-yl)-2-(methylsulfonyl)acetamide |
- |
683247 |
| 3.4.21.42 | 0.000014 |
- |
N-(3'-[[5-carbamimidoyl-2-(methylsulfanyl)thiophen-3-yl]sulfonyl]-6-methylbiphenyl-2-yl)-4-(methylsulfonyl)butanamide |
- |
683247 |
| 3.4.21.42 | 0.000018 |
- |
PEG-linked bis(N-[6-amino-5-[(4-carbamimidamido-3'-[[5-carbamimidoyl-2-(methylsulfanyl)thiophen-3-yl]sulfonyl]-6-methylbiphenyl-2-yl)amino]hept-6-en-1-yl]-6-[[(4-carbamimidamido-3'-[[5-carbamimidoyl-2-(methylsulfanyl)thiophen-3-yl]sulfanyl]biphenyl-2-yl)carbamoyl]amino]hexanamide) |
pH and temperature not specified in the publication |
731435 |
| 3.4.21.42 | 0.00002 |
- |
4-[(2-amino-6-methylphenyl)sulfonyl]-5-(methylsulfanyl)thiophene-2-carboximidamide |
- |
683247 |
| 3.4.21.42 | 0.000022 |
- |
6-[[(3'-[[5-carbamimidoyl-2-(methylsulfanyl)thiophen-3-yl]sulfonyl]-6-methylbiphenyl-2-yl)carbamoyl]amino]hexanoic acid |
- |
683247 |
| 3.4.21.42 | 0.000029 |
- |
PEG-linked tetrakis(4-[[4'-carbamimidamido-2'-(carbamoylamino)biphenyl-3-yl]sulfanyl]-5-(methylsulfanyl)thiophene-2-carboximidamide) |
pH and temperature not specified in the publication |
731435 |
| 3.4.21.42 | 0.00003 |
- |
4-[(2'-methylbiphenyl-3-yl)sulfonyl]-5-(methylsulfanyl)thiophene-2-carboximidamide |
- |
683247 |
| 3.4.21.42 | 0.00003 |
- |
4-[(2'-methylbiphenyl-3-yl)sulfonyl]-5-(methylsulfanyl)thiophene-2-carboximidamide |
pH and temperature not specified in the publication |
731435 |
| 3.4.21.42 | 0.000039 |
- |
PEG-linked bis(6-[[(4-carbamimidamido-3'-[[5-carbamimidoyl-2-(methylsulfanyl)thiophen-3-yl]sulfonyl]-6-methylbiphenyl-2-yl)carbamoyl]amino]hexanamide) |
pH and temperature not specified in the publication |
731435 |
