EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.4.21.22 | -999 |
- |
more |
inhibition kinetics |
683625 |
3.4.21.22 | 0.0000006 |
- |
(7S)-2-methyl-7-phenyl-7-[4-(4H-1,2,4-triazol-4-yl)benzamido]-6,7,8,9-tetrahydropyrido[1,2-a]indole-10-carboxylic acid |
pH and temperature not specified in the publication |
752982 |
3.4.21.22 | 0.0000006 |
- |
(7S)-7-[2-chloro-4-(3-methyl-1H-1,2,4-triazol-1-yl)benzamido]-2-methyl-7-phenyl-6,7,8,9-tetrahydropyrido[1,2-a]indole-10-carboxylic acid |
pH and temperature not specified in the publication |
752982 |
3.4.21.22 | 0.0000008 |
- |
(2E)-3-[(7S)-7-[2-chloro-4-(4H-1,2,4-triazol-4-yl)benzamido]-2-methyl-7-phenyl-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl]prop-2-enoic acid |
pH and temperature not specified in the publication |
752982 |
3.4.21.22 | 0.0000012 |
- |
(7S)-7-[2-chloro-4-(4H-1,2,4-triazol-4-yl)benzamido]-2-methyl-7-phenyl-6,7,8,9-tetrahydropyrido[1,2-a]indole-10-carboxamide |
pH and temperature not specified in the publication |
752982 |
3.4.21.22 | 0.0000016 |
- |
N-[(7S)-10-(5-aminopyridin-3-yl)-2-methyl-7-phenyl-6,7,8,9-tetrahydropyrido[1,2-a]indol-7-yl]-2-chloro-4-(4H-1,2,4-triazol-4-yl)benzamide |
pH and temperature not specified in the publication |
752982 |
3.4.21.22 | 0.0000018 |
- |
2,6-dichloro-N-[(2R)-8-methyl-2-(3-methylphenyl)-1,2,3,4-tetrahydropyrido[1,2-b]indazol-2-yl]-4-(3-methyl-1H-1,2,4-triazol-1-yl)benzamide |
pH and temperature not specified in the publication |
752982 |
3.4.21.22 | 0.000002 |
- |
2-[(2-carbamimidoyl-1-benzothiophen-4-yl)oxy]-2-phenylethyl (2-[[(2-methylpropyl)amino]methyl]phenyl)carbamate |
pH and temperature not specified in the publication |
717964 |
3.4.21.22 | 0.0000021 |
- |
2-chloro-N-[(2R)-8-methyl-2-phenyl-1,2,3,4-tetrahydropyrido[1,2-b]indazol-2-yl]-4-(3-methyl-1H-1,2,4-triazol-1-yl)benzamide |
pH and temperature not specified in the publication |
752982 |
3.4.21.22 | 0.0000024 |
- |
2-chloro-N-[(7S)-10-[(E)-(hydroxyimino)methyl]-2-methyl-7-phenyl-6,7,8,9-tetrahydropyrido[1,2-a]indol-7-yl]-4-(4H-1,2,4-triazol-4-yl)benzamide |
pH and temperature not specified in the publication |
752982 |