EC Number   |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
|---|
   3.2.1.114 | -999 |
- |
more |
although too weak for full Ki analyses with the amounts of material available, all analogues with salacinol-like stereochemistry at positions 2 and 3 proved to be weak inhibitors of the enzyme with IC50 values of approximately 7.5 mM |
666958 |
| 3.2.1.114 | 0.0000105 |
- |
swainsonine |
pH 5.75, 37°C |
646602 |
| 3.2.1.114 | 0.00002 |
- |
(1S,2R,8R,8aR)-octahydroindolizine-1,2,8-triol |
20C, pH 6.8 |
696732 |
| 3.2.1.114 | 0.00002 |
- |
swainsonine |
- |
696214, 696732 |
| 3.2.1.114 | 0.00002 |
- |
swainsonine |
pH 5.6 |
696214 |
| 3.2.1.114 | 0.000036 |
- |
Mannostatin A |
- |
665311, 697318 |
| 3.2.1.114 | 0.000076 |
- |
(1R,2R,3R,4S,5R)-4-amino-5-methoxycyclopentane-1,2,3-triol |
- |
697318 |
| 3.2.1.114 | 0.000135 |
- |
(2S,3R,4S)-2-([[(1R)-2-hydroxy-1-phenylethyl]amino]methyl)pyrrolidine-3,4-diol |
- |
696732 |
| 3.2.1.114 | 0.00015 |
- |
mannostatin B |
- |
697318 |
| 3.2.1.114 | 0.000155 |
- |
swainsonine |
- |
696732 |
