EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
2.7.4.14 | 0.0012 |
- |
P1,P5-di(adenosine-5') pentaphosphate |
versus ATP |
645153 |
2.7.4.14 | 0.00653 |
- |
P1,P5-di(adenosine-5') pentaphosphate |
versus UMP |
645153 |
2.7.4.14 | 0.016 |
- |
5-Cl-uracil vinylphosphonate |
- |
673598 |
2.7.4.14 | 0.017 |
- |
5-Br-uracil vinylphosphonate |
- |
673598 |
2.7.4.14 | 0.028 |
- |
5-Phe-S-uracil vinylphosphonate |
- |
673598 |
2.7.4.14 | 0.12 |
- |
CMP |
pH 7.4, 37°C, GST fusion UMP/CMP kinase |
645162 |
2.7.4.14 | 0.5 |
- |
CMP |
pH 7.4, 37°C, His-tagged UMP/CMP kinase |
645162 |
2.7.4.14 | 0.5 |
- |
UMP |
pH 7.4, 37°C, GST fusion UMP/CMP kinase |
645162 |
2.7.4.14 | 0.7 |
- |
uracil vinylphosphonate |
- |
673598 |
2.7.4.14 | 1.5 |
- |
UMP |
pH 7.4, 37°C, His-tagged UMP/CMP kinase |
645162 |