EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
2.1.1.28 | -999 |
- |
more |
- |
639435, 639436 |
2.1.1.28 | -999 |
- |
more |
enzyme kinetics using competitive tight-binding inhibition routine |
699423 |
2.1.1.28 | 0.000001 |
- |
N-(4-chlorophenyl)-3-(fluoromethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide |
pH 8.0, 30°C, mutant G57A |
699423 |
2.1.1.28 | 0.0000013 |
- |
N-(4-chlorophenyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide |
pH 8.0, 30°C, mutant G57A |
699423 |
2.1.1.28 | 0.0000014 |
- |
N-(4-chlorophenyl)-3-(hydroxymethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide |
pH 8.0, 30°C, mutant G57A |
699423 |
2.1.1.28 | 0.00000155 |
- |
SKF 64139 |
wild type enzyme, inhibition assay containing a fixed concentration of S-adenosyl-L-methionine and variable concentrations of the inhibitor and phenylethanolamine |
675288 |
2.1.1.28 | 0.0000016 |
- |
7,8-dichloro-1,2,3,4-tetrahydroisoquinoline |
pH 8.0, 30°C |
733211 |
2.1.1.28 | 0.0000018 |
- |
3-(fluoromethyl)-7-(thiomorpholin-4-ylsulfonyl)-1,2,3,4-tetrahydroisoquinoline |
pH 8.0, 30°C, mutant G57A |
699423 |
2.1.1.28 | 0.0000031 |
- |
7,8-dichloro-1,2,3,4-tetrahydroisoquinoline |
pH 8.0 |
661339 |
2.1.1.28 | 0.0000031 |
- |
7,8-dichloro-1,2,3,4-tetrahydroisoquinoline |
pH 8.0, 37°C |
696719 |