EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
1.14.16.2 | -999 |
- |
more |
inhibition kinetics |
688519 |
1.14.16.2 | -999 |
- |
more |
value dependent on electron donor, overview |
438693 |
1.14.16.2 | 0.001 |
- |
6-[2-(4-benzoylphenyl)propionyloxymethyl]-5,6,7,8-tetrahydropterin |
- |
438710 |
1.14.16.2 | 0.011 |
- |
3-iodo-L-tyrosine |
versus tetrahydrobiopterin |
438693 |
1.14.16.2 | 0.016 |
- |
2,4-diamino-6-dihydroxypropyl-5,6,7,8-tetrahydropterin |
- |
438710 |
1.14.16.2 | 0.024 |
- |
3-iodo-L-tyrosine |
versus tyrosine, in presence of tetrahydrobiopterin |
438693 |
1.14.16.2 | 0.037 |
- |
L-tyrosine |
pH 7.0, 30°C, mutant enzyme T283M |
660477 |
1.14.16.2 | 0.044 |
- |
L-tyrosine |
pH 7.0, 30°C, mutant enzyme T463M |
660477 |
1.14.16.2 | 0.046 |
- |
L-tyrosine |
pH 7.0, 30°C, wild-type enzyme |
660477 |
1.14.16.2 | 0.048 |
- |
L-tyrosine |
pH 7.0, 30°C, mutant enzyme R306H |
660477 |