EC Number   |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
|---|
    1.1.1.86 | -999 |
- |
1-cyano-N-(4-methylphenyl)cyclopropanecarboxamide |
value above 300 |
685577 |
| 1.1.1.86 | -999 |
- |
more |
- |
639172, 639175 |
| 1.1.1.86 | -999 |
- |
more |
inhibition mechanism and kinetics |
670612 |
| 1.1.1.86 | 0.0000079 |
- |
N-isopropyloxalyl hydroxamate |
pH 8.0, 25°C |
762924 |
| 1.1.1.86 | 0.0000079 |
- |
N-isopropyloxalyl hydroxamate |
pH 8.0, 25°C, intact N-isopropyloxalyl hydroxamate is present in only 25% of binding sites, whereas its deoxygenated form is present in the remaining sites. This deoxy form of N-isopropyloxalyl hydroxamate binds rapidly to the enzyme, but with much weaker affinity (Ki: 0.021 mM) |
762924 |
| 1.1.1.86 | 0.00002 |
- |
1-aminocarbonyl-cyclopropane carboxylate |
- |
686070 |
| 1.1.1.86 | 0.0000222 |
- |
MMV688271 |
pH 8.0, temperature not specified in the publication |
762928 |
| 1.1.1.86 | 0.000026 |
- |
N-Hydroxy-N-isopropyloxamate |
pH 8.0, 25°C |
762676 |
| 1.1.1.86 | 0.0000384 |
- |
MMV688271 |
pH 8.0, temperature not specified in the publication |
762928 |
| 1.1.1.86 | 0.000058 |
- |
1-cyano-cyclopropane carboxylate |
- |
686070 |
