EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
5.4.99.5 | 0.034 |
- |
tyrosine |
70°C, pH 7.6 |
649515 |
5.4.99.5 | 0.00032 |
- |
(1S,3R,5R)-1-hydroxy-5-nitro-2-oxabicyclo[3.3.1]non-6-ene-3-carboxylic acid |
30°C, pH 7.5, wild-type |
651595 |
5.4.99.5 | 0.001 |
- |
(1R,3R,5S)-3-carboxy-1-hydroxy-2-oxabicyclo[3.3.1]non-6-ene-5-carboxylate |
30°C, pH 7.5, wild-type |
651595 |
5.4.99.5 | 0.0023 |
- |
(1R,3R,5S)-3-carboxy-1-hydroxy-2-oxabicyclo[3.3.1]non-6-ene-5-carboxylate |
30°C, pH 7.5, chorismate mutase domain of P-protein |
651595 |
5.4.99.5 | 0.0029 |
- |
(1S,3R,5R)-1-hydroxy-5-nitro-2-oxabicyclo[3.3.1]non-6-ene-3-carboxylic acid |
30°C, pH 7.5, mutant DELTA117-127 |
651595 |
5.4.99.5 | 0.0076 |
- |
(1S,3R,5R)-1-hydroxy-5-nitro-2-oxabicyclo[3.3.1]non-6-ene-3-carboxylic acid |
30°C, pH 7.5, chorismate mutase domain of P-protein |
651595 |
5.4.99.5 | 0.051 |
- |
(1R,3R,5S)-3-carboxy-1-hydroxy-2-oxabicyclo[3.3.1]non-6-ene-5-carboxylate |
30°C, pH 7.5, mutant DELTA117-127 |
651595 |
5.4.99.5 | 0.23 |
- |
(1S,3S,5R)-1-hydroxy-5-nitro-2-oxabicyclo[3.3.1]non-6-ene-3-carboxylic acid |
30°C, pH 7.5, wild-type |
651595 |
5.4.99.5 | 0.0028 |
- |
chorismate |
30°C, pH 7.6, in presence of 0.005 mM tyrosine |
651936 |
5.4.99.5 | -999 |
- |
oxabicyclic dicarboxylic acid |
>> 1 mM mutant C88S/R90K |
652061 |