EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
4.6.1.18 | 0.08124 |
- |
(-)-epigallocatechin-3-gallate |
pH 6.0 |
663854 |
4.6.1.18 | 0.229 |
- |
1-(2,5-dideoxy-5-(4-carboxypiperidinyl)-beta-D-threo-pentofuranosyl)thymine |
pH 7.5, 25°C |
717377 |
4.6.1.18 | 0.423 |
- |
1-(2,5-dideoxy-5-pyrrolidin-1-yl-beta-L-erythro-pentofuranosyl)-5-methylpyrimidine-2,4(1H,3H)-dione |
- |
709463 |
4.6.1.18 | 0.179 |
- |
1-(5-deoxy-5-morpholin-4-yl-alpha-L-arabinofuranosyl)pyrimidine-2,4(1H,3H)-dione |
- |
709463 |
4.6.1.18 | 0.172 |
- |
1-(5-deoxy-5-piperidin-1-yl-alpha-L-arabinofuranosyl)pyrimidine-2,4(1H,3H)-dione |
- |
709463 |
4.6.1.18 | 0.203 |
- |
1-(5-deoxy-5-pyrrolidin-1-yl-alpha-L-arabinofuranosyl)pyrimidine-2,4(1H,3H)-dione |
- |
709463 |
4.6.1.18 | 0.077 |
- |
1-(5-deoxy-5-[4-(ethoxycarbonyl)piperidin-1-yl]-alpha-L-arabinofuranosyl)pyrimidine-2,4(1H,3H)-dione |
- |
709463 |
4.6.1.18 | 0.08 |
- |
2',3'-dideoxy-3'-L-serinylamino thymidine |
- |
707728 |
4.6.1.18 | 0.451 |
- |
2',3'-dideoxy-3'-L-tyrosylamino thymidine |
- |
707728 |
4.6.1.18 | 0.103 |
- |
3'-deoxy-3'-[4-(ethoxycarbonyl)piperidin-1-yl] uridine |
- |
664308 |