EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.5.4.4 | -999 |
- |
more |
inhibition kinetics |
688040 |
3.5.4.4 | -999 |
- |
more |
inhibition kinetics of the large and the small isozyme |
667032 |
3.5.4.4 | -999 |
- |
more |
inhibition kinetics of the large isozyme |
667032 |
3.5.4.4 | -999 |
- |
more |
kinetics and thermodynamic effects of inhibitors, QSAR analysis, overview |
688029 |
3.5.4.4 | -999 |
- |
more |
the adenine moiety of inhibitors does not bind to the histidine residues of the active site His238 |
654788 |
3.5.4.4 | 0.00000011 |
- |
(2S,3R)-3-(6-amino-9H-purin-9-yl)-5-[3-(trifluoromethyl)phenyl]pentan-2-ol |
pH 7.0, temperature not specified in the publication |
752963 |
3.5.4.4 | 0.00000025 |
- |
coformycin |
37°C, pH not specified in the publication |
720969 |
3.5.4.4 | 0.00000043 |
- |
5'-methylthiocoformycin |
- |
687290 |
3.5.4.4 | 0.00000079 |
- |
5'-methylthio-2'-deoxycoformycin |
- |
687290 |
3.5.4.4 | 0.00000114 |
- |
erythro-9-(2-hydroxy-3-nonyl)adenine |
pH 7.2, 30°C |
669783 |