EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.5.4.4 | -999 |
- |
more |
the adenine moiety of inhibitors does not bind to the histidine residues of the active site His238 |
654788 |
3.5.4.4 | 0.00007 |
- |
erythro-9-(2-hydroxy-3-nonyl)-adenine |
pH 7.1, 23°C, after preincubation with diethyl dicarbonate |
654788 |
3.5.4.4 | 0.00008 |
- |
erythro-9-(2-hydroxy-3-nonyl)-adenine |
pH 7.1, 23°C |
654788 |
3.5.4.4 | 0.00009 |
- |
diethyl dicarbonate |
pH 7.1, 23°C, in presence of 0.022 mM erythro-9-(2-hydroxy-3-nonyl)-adenine |
654788 |
3.5.4.4 | 0.00011 |
- |
erythro-9-(2-hydroxy-3-nonyl)-3-deazaadenine |
pH 7.1, 23°C, after preincubation with diethyl dicarbonate |
654788 |
3.5.4.4 | 0.00013 |
- |
diethyl dicarbonate |
pH 7.1, 23°C, in presence of 0.03 mM erythro-9-(2-hydroxy-3-nonyl)-3-deazaadenine |
654788 |
3.5.4.4 | 0.00014 |
- |
erythro-9-(2-hydroxy-3-nonyl)-3-deazaadenine |
pH 7.1, 23°C |
654788 |
3.5.4.4 | 0.007 |
- |
1-deazaadenosine |
pH 7.1, 23°C |
654788 |
3.5.4.4 | 0.0074 |
- |
1-deazaadenosine |
pH 7.1, 23°C, after preincubation with diethyl dicarbonate |
654788 |
3.5.4.4 | 0.01 |
- |
diethyl dicarbonate |
pH 7.1, 23°C, in presence of 0.008 mM 1-deazaadenosine |
654788 |