EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.5.4.4 | 0.00000043 |
- |
5'-methylthiocoformycin |
- |
687290 |
3.5.4.4 | 0.00000079 |
- |
5'-methylthio-2'-deoxycoformycin |
- |
687290 |
3.5.4.4 | 0.0000049 |
- |
1-[(R)-4-(5-(3-(4-chlorophenyl)propoxyl)-1-methylindol-3-yl)-1-hydroxy-2-butyl]imidazole-4-carboxamide |
- |
669771 |
3.5.4.4 | 0.0000075 |
- |
1-[(R)-4-(6-(3-benzylureido)indol-1-yl)-1-hydroxy-2-butyl]imidazole-4-carboxamide |
- |
669771 |
3.5.4.4 | 0.0000077 |
- |
1-[(R)-1-hydroxy-4-(6-(5-phenylvalerylamino)indol-1-yl)-2-butyl]imidazole-4-carboxamide |
- |
669771 |
3.5.4.4 | 0.000011 |
- |
1-[(R)-1-hydroxy-4-(6-(3-(1-methylbenzimidazol-2-yl)propionylamino)indol-1-yl)-2-butyl]imidazole-4-carboxamide |
- |
669771 |
3.5.4.4 | 0.000012 |
- |
1-[(R)-1-hydroxy-4-(6-(4-phenylbutoxy)indol-1-yl)-2-butyl]imidazole-4-carboxamide |
- |
669771 |
3.5.4.4 | 0.000013 |
- |
1-[(R)-4-(5-hexyloxy-1-methylindol-3-yl)-1-hydroxy-2-butyl]imidazole-4-carboxamide |
- |
669771 |
3.5.4.4 | 0.000013 |
- |
1-[(R)-4-(6-(3-(4-chlorophenyl)propoxy)indol-1-yl)-1-hydroxy-2-butyl]imidazole-4-carboxamide |
- |
669771 |
3.5.4.4 | 0.000016 |
- |
1-[(R)-1-hydroxy-4-(6-(4-phenylbutyrylamino)indol-1-yl)-2-butyl]imidazole-4-carboxamide |
- |
669771 |