EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.4.22.69 | 0.0013 |
- |
(S)-N-((S)-1-(benzo[d]thiazol-2-yl)-1-oxo-3-((S)-2-oxopyrrolidin-3-yl)propan-2-yl)-2-((E)-3-(3,4-dimethoxyphenyl)acrylamido)-4-methylpentanamide |
enzyme mutant R188I, pH and temperature not specified in the publication |
731748 |
3.4.22.69 | 0.0007 |
- |
(S)-N-((S)-1-(benzo[d]thiazol-2-yl)-1-oxo-3-((S)-2-oxopyrrolidin-3-yl)propan-2-yl)-2-((E)-3-(4-methoxyphenyl)acrylamido)-4-methylpentanamide |
enzyme mutant R188I, pH and temperature not specified in the publication |
731748 |
3.4.22.69 | 0.0000031 |
- |
(S)-N-((S)-1-(benzo[d]thiazol-2-yl)-1-oxo-3-((S)-2-oxopyrrolidin-3-yl)propan-2-yl)-2-((S)-2-(2-(3-(dimethylamino)phenoxy)acetamido)-3-methylbutanamido)-4-methylpentanamide |
enzyme mutant R188I, pH and temperature not specified in the publication |
731748 |
3.4.22.69 | 0.0013 |
- |
(S)-N-((S)-1-(benzo[d]thiazol-2-yl)-1-oxo-3-((S)-2-oxopyrrolidin-3-yl)propan-2-yl)-2-(2-((2-methoxyphenyl)amino)acetamido)-4-methylpentanamide |
enzyme mutant R188I, pH and temperature not specified in the publication |
731748 |
3.4.22.69 | 0.0007 |
- |
(S)-N-((S)-1-(benzo[d]thiazol-2-yl)-1-oxo-3-((S)-2-oxopyrrolidin-3-yl)propan-2-yl)-2-(2-((3-methoxyphenyl)amino)acetamido)-4-methylpentanamide |
enzyme mutant R188I, pH and temperature not specified in the publication |
731748 |
3.4.22.69 | 0.00069 |
- |
(S)-N-((S)-1-(benzo[d]thiazol-2-yl)-1-oxo-3-((S)-2-oxopyrrolidin-3-yl)propan-2-yl)-2-(2-((4-methoxyphenyl)amino)acetamido)-4-methylpentanamide |
enzyme mutant R188I, pH and temperature not specified in the publication |
731748 |
3.4.22.69 | 0.0074 |
- |
(S)-N-((S)-1-(benzo[d]thiazol-2-yl)-1-oxo-3-((S)-2-oxopyrrolidin-3-yl)propan-2-yl)-2-(2-(3-(dimethylamino)phenoxy)acetamido)-4-methylpentanamide |
enzyme mutant R188I, pH and temperature not specified in the publication |
731748 |
3.4.22.69 | 0.00061 |
- |
(S)-N-((S)-1-(benzo[d]thiazol-2-yl)-1-oxo-3-((S)-2-oxopyrrolidin-3-yl)propan-2-yl)-2-(2-(4-hydroxyphenoxy)acetamido)-4-methylpentanamide |
enzyme mutant R188I, pH and temperature not specified in the publication |
731748 |
3.4.22.69 | 0.00042 |
- |
(S)-N-((S)-1-(benzo[d]thiazol-2-yl)-1-oxo-3-((S)-2-oxopyrrolidin-3-yl)propan-2-yl)-2-(2-(4-methoxyphenyl)acetamido)-4-methylpentanamide |
enzyme mutant R188I, pH and temperature not specified in the publication |
731748 |
3.4.22.69 | 0.00061 |
- |
(S)-N-((S)-1-(benzo[d]thiazol-2-yl)-1-oxo-3-((S)-2-oxopyrrolidin-3-yl)propan-2-yl)-2-(3-(4-methoxyphenyl)propanamido)-4-methylpentanamide |
enzyme mutant R188I, pH and temperature not specified in the publication |
731748 |