EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.4.21.27 | -999 |
- |
more |
- |
683682 |
3.4.21.27 | -999 |
- |
more |
competition for platelet binding by the wild-type enzyme and mutants, overview |
683160 |
3.4.21.27 | -999 |
- |
more |
second-order inhibition rate constants, wild-type and mutant enzymes with different inhibitors, overview |
683157 |
3.4.21.27 | 0.00000002 |
- |
methyl [(11S)-11-([(2E)-3-[5-chloro-2-(1H-tetrazol-1-yl)phenyl]prop-2-enoyl]amino)-6-fluoro-2-oxo-1,3,4,10,11,13-hexahydro-2H-5,9:15,12-di(azeno)-1,13-benzodiazacycloheptadecin-18-yl]carbamate |
at 37°C, pH not specified in the publication |
752995 |
3.4.21.27 | 0.0000002 |
- |
3'-[(2S,4R)-6-carbamimidoyl-4-methyl-4-phenyl-1,2,3,4-tetrahydroquinolin-2-yl]-4-carbamoyl-5'-[(3-methylbutanoyl)amino]biphenyl-2-carboxylic acid |
at pH 7.4 and 37°C |
732318 |
3.4.21.27 | 0.0000003 |
- |
trans-N-((S)-1-(4-(3-amino-1H-indazol-6-yl)-5-fluoro-1H-imidazol-2-yl)-2-phenylethyl)-4-(aminomethyl)cyclohexanecarboxamide |
at pH 7.4 and 37°C |
732318 |
3.4.21.27 | 0.00000031 |
- |
trans-N-[(1S)-1-[4-(3-amino-1H-indazol-6-yl)-5-chloro-1H-imidazol-2-yl]-2-phenylethyl]-4-(aminomethyl)cyclohexanecarboxamide |
at 25°C, pH not specified in the publication |
731462 |
3.4.21.27 | 0.00000031 |
- |
trans-N-[(1S)-1-[4-(3-amino-1H-indazol-6-yl)-5-chloro-1H-imidazol-2-yl]-2-phenylethyl]-4-(aminomethyl)cyclohexanecarboxamide |
pH and temperature not specified in the publication |
731466 |
3.4.21.27 | 0.00000032 |
- |
methyl [(11S)-11-([(2E)-3-[5-chloro-2-(1H-tetrazol-1-yl)phenyl]prop-2-enoyl]amino)-2-oxo-1,3,4,10,11,13-hexahydro-2H-5,9:15,12-di(azeno)-1,13-benzodiazacycloheptadecin-18-yl]carbamate |
at 37°C, pH not specified in the publication |
752995 |
3.4.21.27 | 0.00000053 |
- |
methyl [(11S)-11-([(2E)-3-[5-chloro-2-(1H-tetrazol-1-yl)phenyl]prop-2-enoyl]amino)-6-fluoro-2-oxo-1,3,4,10,11,13-hexahydro-2H-15,12-(azeno)-5,9-(metheno)-1,13-benzodiazacycloheptadecin-18-yl]carbamate |
at 37°C, pH not specified in the publication |
752995 |