EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
2.4.1.65 | -999 |
- |
more |
2,3-dihydroxybenzoic acid: above 0.200, presence of MnCl2, overnight (15 h) pre-incubation of compound and enzyme before initiation of the reaction with GDP-fucose, 2,4-dihydroxybenzoic acid: above 0.200, presence of MnCl2, overnight (15 h) pre-incubation of compound and enzyme before initiation of the reaction with GDP-fucose, 3,5-dimethoxy 4-hydroxybenzoic acid: above 0.200, presence of MnCl2, overnight (15 h) pre-incubation of compound and enzyme before initiation of the reaction with GDP-fucose, 3,4-dimethoxybenzoic acid: above 0.200, presence of MnCl2, overnight (15 h) pre-incubation of compound and enzyme before initiation of the reaction with GDP-fucose, 3,4,5-trimethoxybenzoic acid: above 0.200, presence of MnCl2, overnight (15 h) pre-incubation of compound and enzyme before initiation of the reaction with GDP-fucose |
660797 |
2.4.1.65 | 0.00006 |
- |
3,4,5-Trihydroxybenzoic acid |
presence of MnCl2, overnight (15 h) pre-incubation of compound and enzyme before initiation of the reaction with GDP-fucose |
660797 |
2.4.1.65 | 0.0007 |
- |
(-)-epigallocatechin-3-gallate |
presence of MnCl2, overnight (15 h) pre-incubation of compound and enzyme before initiation of the reaction with GDP-fucose |
660797 |
2.4.1.65 | 0.0012 |
- |
ellagic acid |
presence of MnCl2, overnight (15 h) pre-incubation of compound and enzyme before initiation of the reaction with GDP-fucose |
660797 |
2.4.1.65 | 0.0022 |
- |
(-)-epigallocatechin-3-gallate |
60 min assay, no pre-incubation |
660797 |
2.4.1.65 | 0.0022 |
- |
(-)-epigallocatechin-3-gallate |
overnight (15 h) pre-incubation of compound and enzyme before initiation of the reaction with GDP-fucose, MnCl2 omitted in the overnight pre-incubation mixture |
660797 |
2.4.1.65 | 0.0054 |
- |
3,4,5-Trihydroxybenzoic acid |
overnight (15 h) pre-incubation of compound and enzyme before initiation of the reaction with GDP-fucose, MnCl2 omitted in the overnight pre-incubation mixture |
660797 |
2.4.1.65 | 0.008 |
- |
3,4,5-Trihydroxybenzoic acid |
60 min assay, no pre-incubation |
660797 |
2.4.1.65 | 0.008 |
- |
methyl gallate |
presence of MnCl2, overnight (15 h) pre-incubation of compound and enzyme before initiation of the reaction with GDP-fucose |
660797 |
2.4.1.65 | 0.0256 |
- |
unsaturated carba-fucosyl analogon of GDP-fucose |
- |
661341 |