EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
1.5.1.25 | 0.000032 |
- |
3,5-diiodothyronine |
pH 7.2, 37°C |
743354 |
1.5.1.25 | 0.000035 |
- |
3,3',5'-L-triiodothyronine |
pH 7.2, 37°C |
743354 |
1.5.1.25 | 0.000278 |
- |
3,5,3'-triiodothyronine |
with substrate S-(2-aminoethyl)-L-cysteine ketimine, pH 5.0, temperature not specified in the publication |
741580 |
1.5.1.25 | 0.0006 |
- |
L-thyroxine |
pH 7.2, 37°C, recombinant enzyme |
743355 |
1.5.1.25 | 0.00075 |
- |
3,5,3'-L-triiodothyronine |
pH 7.2, 37°C, recombinant enzyme |
743355 |
1.5.1.25 | 0.032 |
- |
3,5-L-diiodothyronine |
pH 7.2, 37°C, recombinant enzyme |
743355 |
1.5.1.25 | 0.035 |
- |
3,3',5'-L-triiodothyronine |
pH 7.2, 37°C, recombinant enzyme |
743355 |
1.5.1.25 | 0.038 |
- |
4,5-dibromopyrrole-2-carboxylate |
pH 7.2, 37°C |
743354 |
1.5.1.25 | 0.313 |
- |
3,5-diiodo-L-tyrosine |
pH 7.2, 37°C |
743354 |
1.5.1.25 | 0.313 |
- |
3,5-diiodo-L-tyrosine |
pH 7.2, 37°C, recombinant enzyme |
743355 |