EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
1.3.98.1 | 0.1 |
- |
Orotate |
- |
390909 |
1.3.98.1 | 0.0045 |
- |
Orotate |
pH 9.0, 37°C |
390910 |
1.3.98.1 | 0.0102 |
- |
Orotate |
pH 8.0 |
390927 |
1.3.98.1 | 0.0237 |
- |
Orotate |
pH 8.5, 70°C |
655517 |
1.3.98.1 | 0.000004 |
- |
1-(4-Chloro-phenyl)-1H-pyrazole-3,5-dicarboxylic acid 5-phenylamide 3-[(pyridin-3-ylmethyl)-amide] |
- |
656459 |
1.3.98.1 | 0.000004 |
- |
N3-benzyl-1-(4-chlorophenyl)-N5-phenyl-1H-pyrazole-3,5-dicarboxamide |
- |
656459 |
1.3.98.1 | 0.000006 |
- |
1-(4-Chloro-phenyl)-1H-pyrazole-3,5-dicarboxylic acid 3-benzylamide 5-[(4-carbamoyl-phenyl)-amide] |
- |
656459 |
1.3.98.1 | 0.000008 |
- |
1-(4-Chloro-phenyl)-1H-pyrazole-3,5-dicarboxylic acid 5-[(4-piperidin-1-yl-phenyl)-amide] 3-[(pyridin-3-ylmethyl)-amide] |
- |
656459 |
1.3.98.1 | 0.000012 |
- |
1-(4-Methoxy-phenyl)-1H-pyrazole-3,5-dicarboxylic acid 5-phenylamide 3-[(pyridin-3-ylmethyl)-amide] |
- |
656459 |
1.3.98.1 | 0.000026 |
- |
1-(4-Methoxy-phenyl)-1H-pyrazole-3,5-dicarboxylic acid 3-benzylamide 5-[[4-(pyrrolidine-1-carbonyl)-phenyl]-amide] |
- |
656459 |