EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.5.4.4 | 0.016 |
- |
purine riboside |
pH 7.5, 25°C |
655734 |
3.5.4.4 | 0.126 |
- |
acetaminophen |
pH 7.5, 27°C |
656388 |
3.5.4.4 | 0.214 |
- |
acetaminophen |
pH 7.5, 37°C |
656388 |
3.5.4.4 | 0.012 |
- |
7,8-dihydro-1-p-methoxybenzyl-6H-6,7-dimethyl-8-propoxyimidazo[4,5-e][1,2,4]-triazepine |
pH 7.0, 25°C |
656467 |
3.5.4.4 | 0.015 |
- |
8-butoxy-7,8-dihydro-1-p-methoxybenzyl-6H-6,7-dimethylimidazo[4,5-e][1,2,4]triazepine |
pH 7.0, 25°C |
656467 |
3.5.4.4 | 0.02 |
- |
7,8-dihydro-8-ethoxy-1-p-methoxybenzyl-6H-6,7-dimethylimidazo[4,5-e][1,2,4]triazepine |
pH 7.0, 25°C |
656467 |
3.5.4.4 | 0.023 |
- |
7,8-dihydro-1-p-methoxybenzyl-8-(2-methoxyethoxy)-6H-6,7-dimethylimidazo[4,5-e][1,2,4]triazepine |
pH 7.0, 25°C |
656467 |
3.5.4.4 | 0.024 |
- |
7,8-dihydro-8-methoxy-1-p-methoxybenzyl-6H-6,7-dimethylimidazo[4,5-e][1,2,4]triazepine |
pH 7.0, 25°C |
656467 |
3.5.4.4 | 0.03 |
- |
7,8-dihydro-8-isopropoxy-1-p-methoxybenzyl-6H-6,7-dimethylimidazo[4,5-e][1,2,4]triazepine |
pH 7.0, 25°C |
656467 |
3.5.4.4 | 0.077 |
- |
7,8-dihydro-1-p-methoxybenzyl-8-(4-methoxybenzyloxy)-6H-6,7-dimethylimidazo[4,5-e][1,2,4]triazepine |
pH 7.0, 25°C |
656467 |