EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.5.3.1 | 0.013 |
- |
S-(2-boronoethyl)-L-cysteine |
N130A mutant |
696307 |
3.5.3.1 | 0.014 |
- |
Nomega-hydroxy-L-arginine |
pH 9.6, 37°C |
669279 |
3.5.3.1 | 0.017 |
- |
2-(5-methyl-2-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)hydrazinecarbothioamide |
at pH 9.5 and 37°C |
733642 |
3.5.3.1 | 0.02 |
- |
Nomega-hydroxy-L-arginine |
at pH 7.0 and 30°C |
733678 |
3.5.3.1 | 0.023 |
- |
Chloroquine |
at pH 6.8 and 37°C |
685856 |
3.5.3.1 | 0.0305 |
- |
propargylglycine |
chitosan-immobilized enzyme, at pH 7.0 and 40°C |
733226 |
3.5.3.1 | 0.0362 |
- |
iodoacetamide |
chitosan-immobilized enzyme, at pH 7.0 and 40°C |
733226 |
3.5.3.1 | 0.041 |
- |
Chloroquine |
at pH 7.4 and 37°C |
685856 |
3.5.3.1 | 0.0442 |
- |
hydroxylamine |
chitosan-immobilized enzyme, at pH 7.0 and 40°C |
733226 |
3.5.3.1 | 0.05 |
- |
L-ornithine |
product inhibition constant, Co2+-activated mutant S230G, pH 7.4, 37°C |
718861 |