EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
2.7.3.2 | 10 |
- |
L-isoleucine |
versus phosphocreatine, pH 7.5, 37°C |
661901 |
2.7.3.2 | 10.25 |
- |
(2Z)-3-butyl-1-phenyl-2-(phenyltellanyl)oct-2-en-1-one |
0.020 mM organotellurium, preincubation time 5 min, phosphocreatine variable, mitochondrial fraction, pH 7.5, 37°C |
722307 |
2.7.3.2 | 10.55 |
- |
(2Z)-3-butyl-1-phenyl-2-(phenyltellanyl)oct-2-en-1-one |
0.005 mM organotellurium, preincubation time 5 min, ADP variable, cytosolic fraction, pH 7.5, 37°C |
722307 |
2.7.3.2 | 14 |
- |
L-valine |
versus phosphocreatine, pH 7.5, 37°C |
661901 |
2.7.3.2 | 15.45 |
- |
(2Z)-3-butyl-1-phenyl-2-(phenyltellanyl)oct-2-en-1-one |
0.020 mM organotellurium, preincubation time 5 min, ADP variable, cytosolic fraction, pH 7.5, 37°C |
722307 |
2.7.3.2 | 16 |
- |
(2Z)-3-butyl-1-phenyl-2-(phenyltellanyl)oct-2-en-1-one |
0.020 mM organotellurium, preincubation time 5 min, phosphocreatine variable, cytosolic fraction, pH 7.5, 37°C |
722307 |
2.7.3.2 | 16 |
- |
L-leucine |
versus phosphocreatine, pH 7.5, 37°C |
661901 |
2.7.3.2 | 16.15 |
- |
(2Z)-3-butyl-1-phenyl-2-(phenyltellanyl)oct-2-en-1-one |
0.020 mM organotellurium, preincubation time 5 min including reduced glutathione (GSH), phosphocreatine variable, mitochondrial fraction, pH 7.5, 37°C |
722307 |
2.7.3.2 | 16.46 |
- |
(2Z)-3-butyl-1-phenyl-2-(phenyltellanyl)oct-2-en-1-one |
0.020 mM organotellurium, preincubation time 5 min including reduced glutathione (GSH), phosphocreatine variable, cytosolic fraction, pH 7.5, 37°C |
722307 |
2.7.3.2 | 21 |
- |
L-isoleucine |
versus ADP, pH 7.5, 37°C |
661901 |