EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
2.7.3.2 | 1.2 |
- |
glycocyamine |
at pH 8.5 and 25°C |
760912 |
2.7.3.2 | 1.22 |
- |
SDS |
in 5 mM glycine-NaOH (pH 9.0), at 25°C |
701768 |
2.7.3.2 | 2.37 |
- |
(2Z)-3-butyl-1-phenyl-2-(phenyltellanyl)oct-2-en-1-one |
0.005 mM organotellurium, preincubation time 5 min, ADP variable, mitochondrial fraction, pH 7.5, 37°C |
722307 |
2.7.3.2 | 2.53 |
- |
(2Z)-3-butyl-1-phenyl-2-(phenyltellanyl)oct-2-en-1-one |
0.005 mM organotellurium, preincubation time 5 min including reduced glutathione (GSH), ADP variable, mitochondrial fraction, pH 7.5, 37°C |
722307 |
2.7.3.2 | 5.02 |
- |
(2Z)-3-butyl-1-phenyl-2-(phenyltellanyl)oct-2-en-1-one |
0.005 mM organotellurium, preincubation time 5 min including reduced glutathione (GSH), ADP variable, cytosolic fraction, pH 7.5, 37°C |
722307 |
2.7.3.2 | 5.46 |
- |
(2Z)-3-butyl-1-phenyl-2-(phenyltellanyl)oct-2-en-1-one |
0.005 mM organotellurium, preincubation time 5 min, phosphocreatine variable, mitochondrial fraction, pH 7.5, 37°C |
722307 |
2.7.3.2 | 5.67 |
- |
(2Z)-3-butyl-1-phenyl-2-(phenyltellanyl)oct-2-en-1-one |
0.020 mM organotellurium, preincubation time 5 min, ADP variable, mitochondrial fraction, pH 7.5, 37°C |
722307 |
2.7.3.2 | 5.78 |
- |
(2Z)-3-butyl-1-phenyl-2-(phenyltellanyl)oct-2-en-1-one |
0.020 mM organotellurium, preincubation time 5 min including reduced glutathione (GSH), ADP variable, mitochondrial fraction, pH 7.5, 37°C |
722307 |
2.7.3.2 | 6.49 |
- |
(2Z)-3-butyl-1-phenyl-2-(phenyltellanyl)oct-2-en-1-one |
0.005 mM organotellurium, preincubation time 5 min, phosphocreatine variable, cytosolic fraction, pH 7.5, 37°C |
722307 |
2.7.3.2 | 7.1 |
- |
(2Z)-3-butyl-1-phenyl-2-(phenyltellanyl)oct-2-en-1-one |
0.020 mM organotellurium, preincubation time 30 min, ADP variable, cytosolic fraction, pH 7.5, 37°C |
722307 |