EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
2.4.1.65 | 0.045 |
- |
propyl gallate |
presence of MnCl2, overnight (15 h) pre-incubation of compound and enzyme before initiation of the reaction with GDP-fucose |
660797 |
2.4.1.65 | 0.0503 |
- |
dGDP |
at pH 4.5 and 37°C |
735774 |
2.4.1.65 | 0.0671 |
- |
carba-fucosyl analogon of GDP-fucose |
- |
661341 |
2.4.1.65 | 0.0779 |
- |
GDP |
at pH 4.5 and 37°C |
735774 |
2.4.1.65 | 0.0807 |
- |
GTP |
at pH 4.5 and 37°C |
735774 |
2.4.1.65 | 0.102 |
- |
GDP-6-amino-beta-L-fucose |
at pH 4.5 and 37°C |
735774 |
2.4.1.65 | 0.115 |
- |
2,5-dihydroxybenzoic acid |
presence of MnCl2, overnight (15 h) pre-incubation of compound and enzyme before initiation of the reaction with GDP-fucose |
660797 |
2.4.1.65 | 0.137 |
- |
3,4-dihydroxybenzoic acid |
presence of MnCl2, overnight (15 h) pre-incubation of compound and enzyme before initiation of the reaction with GDP-fucose |
660797 |
2.4.1.65 | 0.137 |
- |
[1-(beta-L-fucopyranosyl)-1H-1,2,3-triazole-4-yl]methylguanosine diphosphate |
at pH 4.5 and 37°C |
735774 |
2.4.1.65 | 0.186 |
- |
[1-(beta-D-galactopyranosyl)-1H-1,2,3-triazole-4-yl] methylguanosine diphosphate |
at pH 4.5 and 37°C |
735774 |