EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
1.1.1.267 | 0.1794 |
- |
epigallocatechin gallate |
pH 7.0, 37°C, recombinant enzyme, uncompetitive versus NADPH |
762667 |
1.1.1.267 | 0.24 |
- |
4-(N-formyl-N-hydroxy-amino)-butyric acid |
pH 7.5, 37°C |
672538 |
1.1.1.267 | 0.444 |
- |
3-fluoro-1-deoxy-D-xylulose-5-phosphate |
- |
656890 |
1.1.1.267 | 0.63 |
- |
1,2-dideoxy-D-threo-3-hexulose 6-phosphate |
pH 7.8, 37°C, recombinant wild-type enzyme |
671590 |
1.1.1.267 | 0.733 |
- |
4-fluoro-1-deoxy-D-xylulose-5-phosphate |
- |
656890 |
1.1.1.267 | 1.1 |
- |
1-deoxy-D-xylulose 5-phosphate |
pH 7.9, 30°C, recombinant His-tagged enzyme |
674260 |
1.1.1.267 | 2 |
- |
1,1,1-trifluoro-1-deoxy-D-xylulose 5-phosphoric acid |
pH 7.6, 37°C, recombinant enzyme |
675577 |
1.1.1.267 | 2.4 |
- |
[4-(hydroxyamino)-4-oxobutyl]phosphonic acid |
pH 7.5, 37°C |
672538 |
1.1.1.267 | 2.8 |
- |
sulfamic acid 2-(N-formyl-N-hydroxy-amino)-ethyl ester |
pH 7.5, 37°C |
672538 |
1.1.1.267 | 3.4 |
- |
1,1-difluoro-1-deoxy-D-xylulose 5-phosphoric acid |
pH 7.6, 37°C, recombinant enzyme |
675577 |