EC Number |
kcat/KM Value [1/mMs-1] |
kcat/KM Value Maximum [1/mMs-1] |
Substrate |
Reference |
---|
2.1.1.374 | 0.3075 |
- |
3-methyl-1-oxo-2-[3-oxo-3-(pyrrolidin-1-yl)propyl]-1,5-dihydrobenzo[4,5]imidazo[1,2-a]pyridine-4-carbonitrile |
pH 7.4, 37°C, wild-type enzyme |
760066 |
2.1.1.374 | 2 |
- |
3-methyl-1-oxo-2-[3-oxo-3-(pyrrolidin-1-yl)propyl]-1,5-dihydrobenzo[4,5]imidazo[1,2-a]pyridine-4-carbonitrile |
pH 7.4, 37°C, mutant enzyme S140A |
760066 |
2.1.1.374 | 85.1 |
- |
2-heptyl-1-hydroxyquinolin-4(1H)-one |
pH 7.0 30°C |
759185 |
2.1.1.374 | 204.1 |
- |
2-heptyl-1-hydroxyquinolin-4(1H)-one |
pH 7.0 30°C |
759185 |