EC Number |
kcat/KM Value [1/mMs-1] |
kcat/KM Value Maximum [1/mMs-1] |
Substrate |
Reference |
---|
1.1.1.141 | 900 |
- |
prostaglandin E2 |
pH 8.0, 25°C, 10 nM 2-([(6-bromo-4H-imidazo[4,5-b]pyridin-2-yl)sulfanyl]methyl)benzonitrile |
726267 |
1.1.1.141 | 1200 |
- |
prostaglandin E2 |
pH 8.0, 25°C, 10 nM 3-(2,5-dimethyl-1-phenyl-1H-pyrrol-3-yl)-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepine |
726267 |
1.1.1.141 | 1800 |
- |
prostaglandin E2 |
pH 8.0, 25°C, 10 nM 2-([(6-bromo-4H-imidazo[4,5-b]pyridin-2-yl)sulfanyl]methyl)benzonitrile |
726267 |
1.1.1.141 | 2000 |
- |
prostaglandin E2 |
pH 8.0, 25°C, 4 nM 3-(2,5-dimethyl-1-phenyl-1H-pyrrol-3-yl)-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepine |
726267 |
1.1.1.141 | 2100 |
- |
prostaglandin E2 |
pH 8.0, 25°C, 20 nM [1-(3-methylphenyl)-1H-benzimidazol-5-yl](piperidin-1-yl)methanone |
726267 |
1.1.1.141 | 2500 |
- |
prostaglandin E2 |
pH 8.0, 25°C |
726267 |
1.1.1.141 | 2800 |
- |
prostaglandin E2 |
pH 8.0, 25°C, 10 nM [1-(3-methylphenyl)-1H-benzimidazol-5-yl](piperidin-1-yl)methanone |
726267 |