EC Number |
KM Value [mM] |
KM Value Maximum [mM] |
Substrate |
Reference |
---|
3.4.24.B3 | -999 |
- |
2-[5-Amino-2-(4-fluoro-phenyl)-6-oxo-6H-pyrimidin-1-yl]-N-(1-benzyl-2-oxo-2-thiazol-2-yl-ethyl)-acetamide |
substrate specificity with synthetic substrates |
651898 |
3.4.24.B3 | 0.003 |
- |
dansyl-Pro-Leu-Ala-Leu-Trp-Ala-Arg-NH2 |
pH 6.8, 25°C, mutant Q215R |
649860 |
3.4.24.B3 | 0.0045 |
- |
dansyl-Pro-Leu-Ala-S-[(4-methoxyphenyl)methyl]Cys-Trp-Ala-Arg-NH2 |
pH 6.8, 25°C, mutant Q215L |
649860 |
3.4.24.B3 | 0.0052 |
- |
dansyl-Pro-Leu-Ala-S-[(4-methoxyphenyl)methyl]Cys-Trp-Ala-Arg-NH2 |
pH 6.8, 25°C, wild-type enzyme |
649860 |
3.4.24.B3 | 0.0057 |
- |
dansyl-Pro-Leu-Ala-Leu-Trp-Ala-Arg-NH2 |
pH 6.8, 25°C, mutant Q215Y |
649860 |
3.4.24.B3 | 0.0064 |
- |
dansyl-Pro-Leu-Ala-S-[(4-methoxyphenyl)methyl]Cys-Trp-Ala-Arg-NH2 |
pH 6.8, 25°C, mutant Q215R |
649860 |
3.4.24.B3 | 0.021 |
- |
dansyl-Pro-Leu-Ala-Leu-Trp-Ala-Arg-NH2 |
pH 6.8, 25°C, wild-type enzyme |
649860 |
3.4.24.B3 | 0.088 |
- |
dansyl-Pro-Leu-Ala-Leu-Trp-Ala-Arg-NH2 |
pH 6.8, 25°C, mutant Q215L |
649860 |
3.4.24.B3 | 0.148 |
- |
GGYAELRMGG |
pH 7.5, 37°C, recombinant mutant A235P |
652423 |
3.4.24.B3 | 0.207 |
- |
GGYAELRMGG |
pH 7.5, 37°C |
652423 |