EC Number |
KM Value [mM] |
KM Value Maximum [mM] |
Substrate |
Reference |
---|
3.4.24.15 | -999 |
- |
more |
kinetics of wild-type and mutant TOP |
707401 |
3.4.24.15 | 0.000041 |
- |
7-methoxycoumarin-4-acetyl-[Ala7, Lys(dinitrophenol)9]-bradykinin |
mutant G603A/G604A, 23°C, pH 7.8 |
697880 |
3.4.24.15 | 0.000054 |
- |
7-methoxycoumarin-4-acetyl-[Ala7, Lys(dinitrophenol)9]-bradykinin |
mutant G603A, 23°C, pH 7.8 |
697880 |
3.4.24.15 | 0.000057 |
- |
7-methoxycoumarin-4-acetyl-(L-Ala-L-Lys(2,4-dinitrophenyl))-bradykinin |
pH 7.8, 23°C |
667499 |
3.4.24.15 | 0.000057 |
- |
7-methoxycoumarin-4-acetyl-[Ala7, Lys(dinitrophenol)9]-bradykinin |
wild-type, 23°C, pH 7.8 |
697880 |
3.4.24.15 | 0.00008 |
- |
7-methoxycoumarin-4-acetyl-[Ala7, Lys(dinitrophenol)9]-bradykinin |
mutant Y605F, 23°C, pH 7.8 |
697880 |
3.4.24.15 | 0.00009 |
- |
7-methoxycoumarin-4-acetyl-[Ala7, Lys(dinitrophenol)9]-bradykinin |
mutant G604A, 23°C, pH 7.8 |
697880 |
3.4.24.15 | 0.000129 |
- |
7-methoxycoumarin-4-acetyl-[Ala7, Lys(dinitrophenol)9]-bradykinin |
mutant G599A, 23°C, pH 7.8 |
697880 |
3.4.24.15 | 0.00013 |
- |
7-methoxycoumarin-4-acetyl-(L-Ala-L-Lys(2,4-dinitrophenyl))-bradykinin |
pH 7.8, 23°C, presence of 1.5 M urea |
667499 |
3.4.24.15 | 0.000136 |
- |
7-methoxycoumarin-4-acetyl-[Ala7, Lys(dinitrophenol)9]-bradykinin |
mutant G611A, 23°C, pH 7.8 |
697880 |