EC Number |
Inhibitors |
Structure |
---|
3.5.1.B18 | 1,10-phenanthroline |
25% inhibition at 0.1 mM |
|
3.5.1.B18 | 8-Hydroxyquinoline-5-sulfonate |
complete inhibition at 1 mM |
|
3.5.1.B18 | Cu2+ |
complete inhibition |
|
3.5.1.B18 | DTNB |
25% inhibition at 1 mM |
|
3.5.1.B18 | DTT |
53% inhibition at 1 mM |
|
3.5.1.B18 | EDTA |
21% inhibition at 1 mM |
|
3.5.1.B18 | folate |
substrate inhibition, competitive |
|
3.5.1.B18 | Hg2+ |
complete inhibition |
|
3.5.1.B18 | more |
the enzyme activity is fairly insensitive to serine, cysteine, and aspartic reagents, but is inhibited by metal chelators |
|
3.5.1.B18 | N,N,N',N'-tetrakis[2-pyridylmethyl]ethylenediamine |
i.e. TPEN, 53% inhibition at 0.1 mM |
|