EC Number |
Inhibitors |
Structure |
---|
3.4.21.B34 | Ala-Ala-Phe-chloromethylketone |
500 nM, 90% inhibition |
|
3.4.21.B34 | Asp-Gln-Thr-Gln-Lys-Gln-Tyr-Gln-Glu-Leu-Thr-Phe-Phe-chloromethyl ketone |
- |
|
3.4.21.B34 | benzyloxycarbonyl-Phe-PSI[CO-CONH]Arg-Glu-Phe-OH |
- |
|
3.4.21.B34 | Ca2+ |
100 mM, CaCl2, 57% inhibition |
|
3.4.21.B34 | carbobenzoxy-L-Leu-L-Leu-L-leucinal |
i.e. MG-132, 0.2 mM, 64% inhibition |
|
3.4.21.B34 | decanoyl-Arg-Val-Arg-Lys-chloromethyl ketone |
- |
|
3.4.21.B34 | NEM |
1 mM, enzyme retains 87% of its activity |
|
3.4.21.B34 | tosyl-L-phenylalanine chloromethyl ketone |
- |
|
3.4.21.B34 | tosyl-L-phenylalanine-chloromethylketone |
0.2 mM, 90% inhibition |
|
3.4.21.B34 | Zn2+ |
25 mM ZnCl2, 60% inhibition |
|