EC Number |
Inhibitors |
Structure |
---|
3.4.21.B28 | 1-benzyl-7-(but-2-yn-1-yl)-3-methyl-8-(piperazin-1-yl)-3,7-dihydro-1H-purine-2,6-dione |
- |
|
3.4.21.B28 | 1-[(4-methoxyquinazolin-2-yl)methyl]-3,7-dimethyl-8-(3-oxopiperazin-1-yl)-3,7-dihydro-1H-purine-2,6-dione |
- |
|
3.4.21.B28 | 1-[(4-methoxyquinazolin-2-yl)methyl]-3-methyl-7-(3-methylbut-2-en-1-yl)-8-(3-oxopiperazin-1-yl)-3,7-dihydro-1H-purine-2,6-dione |
- |
|
3.4.21.B28 | 1-[(4-methoxyquinazolin-2-yl)methyl]-3-methyl-7-(4-methylpent-3-en-1-yl)-8-(3-oxopiperazin-1-yl)-3,7-dihydro-1H-purine-2,6-dione |
- |
|
3.4.21.B28 | 2-mercaptoethanol |
inhibition at 140 mM |
|
3.4.21.B28 | 3,7-dimethyl-8-(3-oxopiperazin-1-yl)-3,7-dihydro-1H-purine-2,6-dione |
- |
|
3.4.21.B28 | 3-[[7-(but-2-yn-1-yl)-3-methyl-2,6-dioxo-8-(piperazin-1-yl)-2,3,6,7-tetrahydro-1H-purin-1-yl]methyl]benzonitrile |
- |
|
3.4.21.B28 | 4'-[[7-(but-2-yn-1-yl)-3-methyl-2,6-dioxo-8-(piperazin-1-yl)-2,3,6,7-tetrahydro-1H-purin-1-yl]methyl]biphenyl-2-carbonitrile |
- |
|
3.4.21.B28 | 4-(2-aminoethyl)-benzenesulfonyl fluoride hydrochloride |
AEBSF, inhibition at 5 mM |
|
3.4.21.B28 | 4-(2-aminoethyl)-benzenesulfonylfluoride |
5 mM |
|