EC Number |
Inhibitors |
Structure |
---|
3.4.21.4 | (2R,4R)-4-phenyl-1-[Nalpha-(7-methoxy-2-naphthalenesulfonyl)-L-arginyl]-2-piperidinecarboxylic acid |
competitive, small molecular weight inhibitor without tryptase inhibitor activity |
|
3.4.21.4 | (4-(6-chloro-naphthalene-2-sulfonyl)-piperazin-1-yl)-(3,4,5-6-tetrahydro[2H-1,4']bipyridinyl-4yl)-methanone |
- |
|
3.4.21.4 | 1,10-phenanthroline |
- |
|
3.4.21.4 | 1-(L-trans-epoxysuccinyl-leucylamino)-4-guanidinobutane |
6.09% inhibition at 0.1 mM |
|
3.4.21.4 | 1-(L-trans-epoxysuccinyl-leucylamino)-4-guanidinobutane |
16.9% inhibition at 0.1 mM |
|
3.4.21.4 | 1-[N2-[(7-methoxynaphthalen-2-yl)sulfonyl]-L-arginyl]-4-phenylpiperidine-2-carboxylic acid |
IC50: 0.0003 mM |
|
3.4.21.4 | 2,7-bis(4-amidinobenzylidene)-cycloheptan-1-one |
- |
|
3.4.21.4 | 2,7-bis(4-amidinobenzylidene)cycloheptan-1-one |
unspecific strong inhibition |
|
3.4.21.4 | 2-mercaptoethanol |
0.1 mM, isoenzyme aT-I loses 90% of its activity, isoenzyme aT-II loses 93% of its activity |
|
3.4.21.4 | 3,4-dichloroisocoumarin |
- |
|