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Results 1 - 10 of 81 > >>
EC Number Inhibitors Commentary Structure
Show all pathways known for 2.7.7.3Display the word mapDisplay the reaction diagram Show all sequences 2.7.7.3(1S,2S)-N-(3,4-dichlorobenzyl)-2-(4,6-dimethoxypyrimidin-2-yl)cyclohexanecarboxamide - Go to the Ligand Summary Page
Show all pathways known for 2.7.7.3Display the word mapDisplay the reaction diagram Show all sequences 2.7.7.3(1S,2S)-N-(3-chlorobenzyl)-2-(4,6-dimethoxypyrimidin-2-yl)cyclohexanecarboxamide - Go to the Ligand Summary Page
Show all pathways known for 2.7.7.3Display the word mapDisplay the reaction diagram Show all sequences 2.7.7.3(2'R)-1-methyl-N4'-[3-(trifluoromethyl)phenyl]-1,2-dihydro-5'H-spiro[indole-3,2'-[1,3,5]triazine]-4',6'-diamine identified by virtual screening. Compound directly binds and blocks access of substrates to the active site. The trifluoromethyl group of the ligand is oriented inside the protein molecule. One of the nitrogen atoms of the ligand forms contacts with Gly8 and Ser9. The NH2 interacts with the guanidine group of Arg90 Go to the Ligand Summary Page
Show all pathways known for 2.7.7.3Display the word mapDisplay the reaction diagram Show all sequences 2.7.7.3(2S)-2-(3-chlorophenyl)-2-[(5-methyl-7-oxo-4,7-dihydro[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)amino]ethyl carbamate - Go to the Ligand Summary Page
Show all pathways known for 2.7.7.3Display the word mapDisplay the reaction diagram Show all sequences 2.7.7.3(3R)-3-(3-chlorophenyl)-3-[(5-methyl-1H-imidazo[4,5-b]pyridin-2-yl)amino]propanenitrile - Go to the Ligand Summary Page
Show all pathways known for 2.7.7.3Display the word mapDisplay the reaction diagram Show all sequences 2.7.7.3(3R)-3-(3-chlorophenyl)-3-[(5-methyl-4,7-dihydro[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)amino]propanenitrile lead compound as selective, small molecule inhibitor, displays modest cellular potency against the efflux-deficient Escherichia coli DeltatolC mutant strain Go to the Ligand Summary Page
Show all pathways known for 2.7.7.3Display the word mapDisplay the reaction diagram Show all sequences 2.7.7.3(3R)-3-(3-chlorophenyl)-3-[(5-methyl-4,7-dihydro[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)amino]propanenitrile lead compound as selective, small molecule inhibitor Go to the Ligand Summary Page
Show all pathways known for 2.7.7.3Display the word mapDisplay the reaction diagram Show all sequences 2.7.7.3(3R)-3-(3-chlorophenyl)-3-[(5-methyl-7-oxo-4,7-dihydro[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)amino]propanenitrile lead compound as selective, small molecule inhibitor, displays modest cellular potency against the efflux-deficient Escherichia coli DeltatolC mutant strain Go to the Ligand Summary Page
Show all pathways known for 2.7.7.3Display the word mapDisplay the reaction diagram Show all sequences 2.7.7.3(3R)-3-(3-chlorophenyl)-3-[(5-methyl-7-oxo-4,7-dihydro[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)amino]propanenitrile lead compound as selective, small molecule inhibitor Go to the Ligand Summary Page
Show all pathways known for 2.7.7.3Display the word mapDisplay the reaction diagram Show all sequences 2.7.7.3(3R)-3-(3-chlorophenyl)-3-[(7-[[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]amino]-5-methyl-1H-imidazo[4,5-b]pyridin-2-yl)amino]propanenitrile - Go to the Ligand Summary Page
Results 1 - 10 of 81 > >>