EC Number |
Inhibitors |
Structure |
---|
2.1.1.6 | (-)-epicatechin-3-gallate |
IC50: 0.0002 mM with 2-hydroxyestradiol as substrate, IC50: 0.0003 mM with 4-hydroxyestradiol as substrate |
|
2.1.1.6 | (-)-epigallocatechin |
IC50: 0.044 mM with 2-hydroxyestradiol as substrate, IC50: 0.05 nM with 4-hydroxyestradiol as substrate |
|
2.1.1.6 | (-)-epigallocatechin gallate |
potent inhibitor with epigallocatechin or 3,4-dihydroxy-L-Phe as substrates |
|
2.1.1.6 | (-)-epigallocatechin gallate-4''-O-glucuronide |
with epigallocatechin or 3,4-dihydroxy-L-Phe as substrates |
|
2.1.1.6 | (-)-epigallocatechin gallate-7-O-glucuronide |
with epigallocatechin or 3,4-dihydroxy-L-Phe as substrates |
|
2.1.1.6 | (-)-epigallocatechin-3-gallate |
IC50: 70 nM with 2-hydroxyestradiol as substrate, IC50: 80 nM with 4-hydroxyestradiol as substrate, mixed inhibitor |
|
2.1.1.6 | (-)-epigallocatechin-3-gallate |
- |
|
2.1.1.6 | (-)-epigallocatechin-3-gallate-3''-O-glucuronide |
IC50: 0.002 mM with 2-hydroxyestradiol as substrate, IC50: 0.0025 mM with 4-hydroxyestradiol as substrate |
|
2.1.1.6 | (-)-epigallocatechin-3-gallate-3'-O-glucuronide |
IC50: 0.0018 mM with 2-hydroxyestradiol as substrate, IC50: 0.0023 mM with 4-hydroxyestradiol as substrate |
|
2.1.1.6 | (-)-epigallocatechin-3-gallate-4''-O-glucuronide |
IC50: 0.0025 mM with 2-hydroxyestradiol as substrate, IC50: 0.004 mM with 4-hydroxyestradiol as substrate |
|