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Results 1 - 10 of 31 > >>
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EC Number Inhibitors Commentary Structure
Show all pathways known for 1.5.3.13Display the word mapDisplay the reaction diagram Show all sequences 1.5.3.131,12-diaminododecane 1,12-diaminododecane derivatives could represent good candidates for the development of novel highly specific mPAO inhibitors Go to the Ligand Summary Page
Show all pathways known for 1.5.3.13Display the word mapDisplay the reaction diagram Show all sequences 1.5.3.131,8-diaminooctane competitive versus the polyamine Go to the Ligand Summary Page
Show all pathways known for 1.5.3.13Display the word mapDisplay the reaction diagram Show all sequences 1.5.3.136,6'-[ethane-1,2-diyldi(piperidine-4,1-diyl)]bis[N-[(2-methoxyphenyl)methyl]hexan-1-amine] 17fold selectivity for spermine oxidase over polyamine oxidase Go to the Ligand Summary Page
Show all pathways known for 1.5.3.13Display the word mapDisplay the reaction diagram Show all sequences 1.5.3.13Chlorhexidine - Go to the Ligand Summary Page
Show all pathways known for 1.5.3.13Display the word mapDisplay the reaction diagram Show all sequences 1.5.3.13guazatine - Go to the Ligand Summary Page
Show all pathways known for 1.5.3.13Display the word mapDisplay the reaction diagram Show all sequences 1.5.3.13MDL72527 - Go to the Ligand Summary Page
Show all pathways known for 1.5.3.13Display the word mapDisplay the reaction diagram Show all sequences 1.5.3.13MDL72527 irreversible. In addition to the covalent adduct, a second MDL72527 molecule is bound in the active site. Binding of MDL72527 is accompanied by altered conformations in the APAO backbone Go to the Ligand Summary Page
Show all pathways known for 1.5.3.13Display the word mapDisplay the reaction diagram Show all sequences 1.5.3.13methoctramine 120fold selectivity for spermine oxidase over polyamine oxidase Go to the Ligand Summary Page
Show all pathways known for 1.5.3.13Display the word mapDisplay the reaction diagram Show all sequences 1.5.3.13more no inhibition at pH 7.5: 1,8-diaminooctane. Comparative study on murine PAO (mPAO) and SMO (mSMO) inhibition. The different behaviour displayed by 1,12-diaminododecane towards mPAO and mSMO reveals the occurrence of basic differences in the ligand binding mode of the two enzymes, the first enzyme interacting mainly with substrate secondary amino groups and the second one with substrate primary amino groups. The data provide the basis for the development of novel and selective inhibitors able to discriminate between mammalian SMO and PAO activities Go to the Ligand Summary Page
Show all pathways known for 1.5.3.13Display the word mapDisplay the reaction diagram Show all sequences 1.5.3.13more no inhibitory activity: N-(3-aminopropyl)-N-2-propynyl-1,4-butanediamine and N-[3-(2-propynylamino)propyl]-1,4-butanediamine Go to the Ligand Summary Page
Results 1 - 10 of 31 > >>
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