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Results 1 - 10 of 10
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EC Number Inhibitors Commentary Structure
Show all pathways known for 5.1.3.13Display the word mapDisplay the reaction diagram Show all sequences 5.1.3.131-(3-(5-allyl-5H-[1,2,4]triazino[5,6-b]indol-3-ylsulfonyl)-propyl)-1H-benzo[d]imidazol-2(3H)-one - Go to the Ligand Summary Page
Show all pathways known for 5.1.3.13Display the word mapDisplay the reaction diagram Show all sequences 5.1.3.131-(3-(5-allyl-5H-[1,2,4]triazino[5,6-b]indol-3-ylthio)propyl)-1H-benzo[d]imidazol-2(3H)-one i.e. 77074, a SID 7975595 analogue Go to the Ligand Summary Page
Show all pathways known for 5.1.3.13Display the word mapDisplay the reaction diagram Show all sequences 5.1.3.131-(3-(5-allyl-8-methyl-5H-[1,2,4]triazino[5,6-b]indol-3-ylthio)propyl)-1H-benzo[d]imidazol-2(3H)-one - Go to the Ligand Summary Page
Show all pathways known for 5.1.3.13Display the word mapDisplay the reaction diagram Show all sequences 5.1.3.131-(3-(5-ethyl-5H-[1,2,4]triazino[5,6-b]indol-3-ylsulfonyl)-propyl)-1H-benzo[d]imidazol-2(3H)-one - Go to the Ligand Summary Page
Show all pathways known for 5.1.3.13Display the word mapDisplay the reaction diagram Show all sequences 5.1.3.131-(3-(5-ethyl-5H-[1,2,4]triazino[5,6-b]indol-3-ylthio)propyl)-1H-benzo[d]imidazol-2(3H)-one i.e. SID 7975595, a competitive, fast-on rate, fully reversible inhibitor of RmlC. Increases the Km for TDP-6-deoxy-D-xylo-hexopyranosid-4-ulose. Cytotoxic SID 7975595 has an IC50 of approximately 0.075 mM in HAE cells Go to the Ligand Summary Page
Show all pathways known for 5.1.3.13Display the word mapDisplay the reaction diagram Show all sequences 5.1.3.131-(3-(5-methyl-5H-[1,2,4]triazino[5,6-b]indol-3-ylthio)propyl)-1H-benzo[d]imidazol-2(3H)-one i.e. 77072, a SID 7975595 analogue Go to the Ligand Summary Page
Show all pathways known for 5.1.3.13Display the word mapDisplay the reaction diagram Show all sequences 5.1.3.131-(3-(5-methylphenyl-5H-[1,2,4]triazino[5,6-b]indol-3-ylthio)propyl)-1H-benzo[d]imidazol-2(3H)-one i.e. 77070, a SID 7975595 analogue Go to the Ligand Summary Page
Show all pathways known for 5.1.3.13Display the word mapDisplay the reaction diagram Show all sequences 5.1.3.131-(3-(5-propyl-5H-[1,2,4]triazino[5,6-b]indol-3-ylthio)propyl)-1H-benzo[d]imidazol-2(3H)-one i.e. 77071, a SID 7975595 analogue Go to the Ligand Summary Page
Show all pathways known for 5.1.3.13Display the word mapDisplay the reaction diagram Show all sequences 5.1.3.131-(3-(5H-[1,2,4]triazino[5,6-b]indol-3-ylthio)propyl)-1H-benzo[d]imidazol-2(3H)-one i.e. 77073, a SID 7975595 analogue Go to the Ligand Summary Page
Show all pathways known for 5.1.3.13Display the word mapDisplay the reaction diagram Show all sequences 5.1.3.13more modeling of triazinoindol-benzimidazolones into the active site of RmlC, overview Go to the Ligand Summary Page
Results 1 - 10 of 10
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