Any feedback?
Please rate this page
(search_result.php)
(0/150)

BRENDA support

Refine search

Search Inhibitors

show results
Don't show organism specific information (fast!)
Search organism in taxonomic tree (slow, choose "exact" as search mode, e.g. "mammalia" for rat,human,monkey,...)
(Not possible to combine with the first option)
Refine your search
Image of 2D Structure
Search for synonyms (with exact matching search term)

Search term:

Results 1 - 10 of 299 > >>
EC Number Inhibitors Commentary Structure
Display the word mapDisplay the reaction diagram Show all sequences 3.4.22.51more pro-region of the trypanosomal enzyme inhibits the enzyme function, cystatins and kininogens are inhibitors, overview: inhibitors Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 3.4.22.51more in general immunoglobulin G fractions isolated from rabbits immunised with rabbit apha2-macroglobulin-recombinant catalytic domain of congopain-complexes are the most inhibitory towards the proteolytic activity of congopain. Antibodies produced by rabbits immunised with recombinant catalytic domain of congopain in Freund's adjuvant are generally found to weakly inhibit congopain with a maximum of 40% Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 3.4.22.51more synthesis of 2-hydrazolyl-4-thiazolidinones based on multicomponent reactions and biological evaluation against Trypanosoma cruzi, inhibitory potencies and cytotoxic effects, molecular modeling and QSAR studies, overview. No inhibition by (RS)-2-(2-(2-bromobenzylidene)hydrazono)-3-methyl-4-oxo-5-thiazolidine-N-methylacetamide and (Z)-((2-(4-fluorobenzylidene)hydrazono)-3-methyl-5-methoxycarbonylmethylene)thiazolidin-4-one at 0.1 mM Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 3.4.22.51more synthesis and inhibitory effects against cruzipaon of a series of thirty-three chalcone and seven hydrazide derivatives, overview Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 3.4.22.51more AM1 semi-empirical molecular modeling studies analysing cruzain inhibitory activity, overview Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 3.4.22.51more 0.01% (v/v) of Triton X-100 does not interfere with enzyme activity Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 3.4.22.51more not inhibited by CA-074-OMe Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 3.4.22.51more the AS2 site as a target for the design of cruzain inhibitors is limited Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 3.4.22.51more apolar substituents or halogen atom substitution at the aryl position improved cruzain inhibition and antiparasitic activity in comparison to unsubstituted thiosemicarbazone Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 3.4.22.51more nitrile-based inhibitors are efficient inhibitors of cruzain that bind by forming a covalent bond with this enzyme Go to the Ligand Summary Page
Results 1 - 10 of 299 > >>