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Results 1 - 10 of 13 > >>
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EC Number Inhibitors Commentary Structure
Display the word mapDisplay the reaction diagram Show all sequences 2.4.1.288(1S,2S,3S,4S,5R)-1-[(1S)-1,2-dihydroxyethyl]-4-[[(furan-2-yl)methyl]amino]bicyclo[3.1.0]hexane-2,3-diol UDP-Gal analogue, 82% inhibition at 4 mM Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 2.4.1.288(2R,3R,4R,5R)-2-(2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)-4-hydroxy-5-(hydroxymethyl)tetrahydrofuran-3-yl hydrogen ((E)-((3R,4R,5S)-5-((R)-1,2-dihydroxyethyl)-3,4-dihydroxydihydrofuran-2(3H)-ylidene)fluoromethyl)phosphonate - Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 2.4.1.288(2R,3R,4R,5R)-2-(2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)-4-hydroxy-5-(hydroxymethyl)tetrahydrofuran-3-yl hydrogen ((Z)-((3R,4R,5S)-5-((R)-1,2-dihydroxyethyl)-3,4-dihydroxydihydrofuran-2(3H)-ylidene)fluoromethyl)phosphonate - Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 2.4.1.288(3S,4S)-3-(1,2-dihydroxyethyl)-4-hydroxy-1-(2-phenylethyl)tetrahydrothiophenium chloride sulfonium ion compound as analogue of the donor substrate, uridine diphosphategalactofuranose. The compound contains moieties that mimic both galactofuranose and uridine diphosphate domains, and carries a permanent positive charge to mimic the oxocarbenium ion-like transition state. About 60% inhibition at 4 mM Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 2.4.1.288(3S,4S)-3-(1,2-dihydroxyethyl)-4-hydroxy-1-[2-(4-nitrophenyl)ethyl]tetrahydrothiophenium bromide sulfonium ion compound as analogue of the donor substrate, uridine diphosphategalactofuranose. The compound contains moieties that mimic both galactofuranose and uridine diphosphate domains, and carries a permanent positive charge to mimic the oxocarbenium ion-like transition state. About 50% inhibition at 4 mM Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 2.4.1.2882-[(5E)-5-[(3,4-dichlorophenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-3-yl]-3-(4-iodophenyl)propanoic acid UDP-galactopyranose mutase inhibitor, binding energy value of -8.08 kcal/mol. Compound passes the ADME evaluation and the predicted toxicity evaluation Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 2.4.1.288EDTA - Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 2.4.1.288more not inhibited by UDP-2''-O-methyl-alpha-D-galactofuranose Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 2.4.1.288UDP-3''-deoxy-alpha-D-xylo-hexofuranose 68% inhibition at 1.25 mM Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 2.4.1.288UDP-5''-O-methyl-alpha-D-galactofuranose 15% inhibition at 1.25 mM Go to the Ligand Summary Page
Results 1 - 10 of 13 > >>
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