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<< < Results 11 - 18 of 18
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EC Number Inhibitors Commentary Structure
Display the word mapDisplay the reaction diagram Show all sequences 2.1.1.366N-[[2-(3,5-dimethyl-4H-1,2,4-triazol-4-yl)cyclohexyl]methyl]acetamide SETDB1-TTD inhibitor, binds in the aromatic cage of the Kac pocket of the SETDB1-TTD. It displayed weak binding by SPR and ITC Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 2.1.1.366N2-(3'-[[4-(4-butylpiperazin-1-yl)pyridine-2-carbonyl]amino][1,1'-biphenyl]-4-carbonyl)-6-pyrrolidin-1-yl-L-norleucinamide SETDB1-TTD inhibitor, shows competitive inhibition and docked between the Tudor 2 and 3 Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 2.1.1.366N2-(3'-[[4-(4-butylpiperazin-1-yl)pyridine-2-carbonyl]amino][1,1'-biphenyl]-4-carbonyl)-N6,N6-dimethyl-L-lysinamide SETDB1-TTD inhibitor, shows competitive inhibition and docks between the Tudor 2 and 3 domains Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 2.1.1.366N2-(3'-[[4-(4-methylpiperazin-1-yl)pyridine-2-carbonyl]amino][1,1'-biphenyl]-4-carbonyl)-6-pyrrolidin-1-yl-L-norleucinamide SETDB1-TTD inhibitor, shows competitive inhibition and docks between the Tudor 2 and 3 domains Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 2.1.1.366N2-[3'-[(4-[4-[3-(dimethylamino)propyl]piperazin-1-yl]pyridine-2-carbonyl)amino][1,1'-biphenyl]-4-carbonyl]-6-pyrrolidin-1-yl-L-norleucinamide SETDB1-TTD inhibitor, shows competitive inhibition and docks between the Tudor 2 and 3 domains Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 2.1.1.366N2-[3'-[(4-[4-[3-(dimethylamino)propyl]piperazin-1-yl]pyridine-2-carbonyl)amino][1,1'-biphenyl]-4-carbonyl]-N6,N6-dimethyl-L-lysinamide SETDB1-TTD inhibitor, shows competitive inhibition and docks between the Tudor 2 and 3 domains Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 2.1.1.366N4-[6-(dimethylamino)hexyl]-N2-[5-(dimethylamino)pentyl]-6,7-dimethoxyquinazoline-2,4-diamine SETDB1-TTD inhibitor, shows competitive inhibition and docks between the Tudor 2 and 3 domains Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 2.1.1.366N6,N6-dimethyl-L-lysyl-L-serylthreonyl-N-([4-[2-(acetamidomethyl)cyclohexyl]-4H-1,2,4-triazol-3-yl]methyl)glycinamide - Go to the Ligand Summary Page
<< < Results 11 - 18 of 18
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