5.3.99.2 0.000021 - 2-phenyl-5-(1H-pyrazol-3-yl)-1,3-thiazole 37°C 693542 5.3.99.2 0.000026 - N-[5-(1H-indol-4-yl)pyridin-3-yl]-3-(pyridin-3-yl)propanamide at 37°C, pH not specified in the publication 747270 5.3.99.2 0.000031 - 6-phenoxy-N-[1-(2,2,2-trifluoroethyl)piperidin-4-yl]pyridine-3-carboxamide at 37°C, pH not specified in the publication 747270 5.3.99.2 0.000032 - N-[5-(1H-indol-4-yl)pyridin-3-yl]propanamide at 37°C, pH not specified in the publication 747270 5.3.99.2 0.000035 - N-[5-(1H-indol-4-yl)pyridin-3-yl]-5-oxopyrrolidine-2-carboxamide (incorrect configuration definition!) at 37°C, pH not specified in the publication 747270 5.3.99.2 0.00004 - 3-(3-cyclopropyl-1H-pyrazol-4-yl)-N-ethyl-5,7-dihydro-6H-pyrrolo[3,4-b]pyridine-6-carboxamide pH and temperature not specified in the publication 748543 5.3.99.2 0.000043 - N-[5-(1H-indol-4-yl)pyridin-3-yl]-2-(1H-tetrazol-1-yl)acetamide at 37°C, pH not specified in the publication 747270 5.3.99.2 0.000048 - 6-(piperidin-1-yl)-N-[1-(2,2,2-trifluoroethyl)piperidin-4-yl]pyridine-3-carboxamide at 37°C, pH not specified in the publication 747270 5.3.99.2 0.00006 - 6-(3-methoxyphenyl)-N-[1-(2,2,2-trifluoroethyl)piperidin-4-yl]pyridine-3-carboxamide at 37°C, pH not specified in the publication 747270 5.3.99.2 0.000071 - 6'-oxo-N-[1-(2,2,2-trifluoroethyl)piperidin-4-yl]-1',6'-dihydro[2,2'-bipyridine]-5-carboxamide at 37°C, pH not specified in the publication 747270