3.4.24.B10 0.0000167 - N-[(2E)-3-(3-bromophenyl)-2-[(furan-2-ylcarbonyl)amino]prop-2-enoyl]glycine IC50: 16.7 nM 667947 3.4.24.B10 0.0000248 - N-[(2E)-3-(4-bromofuran-2-yl)-2-[[(5-bromofuran-2-yl)carbonyl]amino]prop-2-enoyl]alanine IC50: 24.8 nM 667947 3.4.24.B10 0.000025 - batimastat with 5-Fam-HALAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C 733079 3.4.24.B10 0.000028 - batimastat with 5-Fam-FFLAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C 733079 3.4.24.B10 0.0000405 - N-[(2E)-3-(2-fluorophenyl)-2-[(phenylcarbonyl)amino]prop-2-enoyl]valine IC50: 40.5 nM 667947 3.4.24.B10 0.0000423 - N-[(2E)-3-furan-2-yl-2-[(furan-2-ylcarbonyl)amino]prop-2-enoyl]alanine IC50: 42.3 nM 667947 3.4.24.B10 0.00012 - MMP inhibitor V with 5-Fam-FFLAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C 733079 3.4.24.B10 0.00018 - MMP inhibitor V with 5-Fam-HALAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C 733079 3.4.24.B10 0.00035 - TAPI-0 with 5-Fam-HALAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C 733079 3.4.24.B10 0.0004 - TAPI-0 with 5-Fam-FFLAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C 733079