2.5.1.9 0.0000013 - N-[2,4-dioxo-6-(ribitylamino)-1,2,3,4-tetrahydropyrimidin-5-yl]oxalamic acid ethyl ester pH 7.0, 27°C 688578 2.5.1.9 0.00235 - 2-[ethyl(methyl)amino]ethyl 4-[(5-ethyl-4-oxo-4,5-dihydrothieno[3,2-c]quinoline-2-carbonyl)amino]benzoate pH 7.5, 37°C 759180 2.5.1.9 0.01912 - ethyl 5-(diethylcarbamoyl)-2-[2-(4-methoxyphenoxy)acetamido]-4-methylthiophene-3-carboxylate pH 7.5, 37°C 759180 2.5.1.9 0.01915 - (2E)-3-(2,3-dimethoxyphenyl)-N-[4-methyl-2-(4-methylpiperazin-1-yl)quinolin-6-yl]prop-2-enamide pH 7.5, 37°C 759180 2.5.1.9 0.02564 - 2-(4-ethoxyphenyl)-N-[3-(piperidin-1-yl)propyl]imidazo[2,1-b][1,3]benzothiazole-7-carboxamide pH 7.5, 37°C 759180 2.5.1.9 0.02638 - N-[3-(azepan-1-yl)propyl]-2-(4-methoxyphenyl)imidazo[2,1-b][1,3]benzothiazole-7-carboxamide pH 7.5, 37°C 759180 2.5.1.9 0.0278 - N-[3-(diethylamino)propyl]-2-(4-ethoxyphenyl)imidazo[2,1-b][1,3]benzothiazole-7-carboxamide pH 7.5, 37°C 759180 2.5.1.9 0.02964 - (2-ethyl-5-oxo-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methyl 3,4,5-triethoxybenzoate pH 7.5, 37°C 759180 2.5.1.9 0.03053 - 5-[3-(propan-2-yl)-1H-pyrazol-5-yl]-3-(3,4,5-trimethoxyphenyl)-1,2,4-oxadiazole pH 7.5, 37°C 759180 2.5.1.9 0.03118 - 2-(4-methoxyphenyl)-N-[3-(piperidin-1-yl)propyl]imidazo[2,1-b][1,3]benzothiazole-7-carboxamide pH 7.5, 37°C 759180