3.1.1.79 0.000001 - morpholin-4-yl-carbamic acid 4-[(4-tert-butyl-cyclohexanecarbonyl)-amino]-phenyl ester IC50: 1 nM 664316 3.1.1.79 0.000002 - (5-chloro-2-[([6-[4-(trifluoromethyl)phenoxy]pyridin-3-yl]carbonyl)amino]phenyl)boronic acid pH 7.3, 37°C 750039 3.1.1.79 0.000003 - (3,4-dihydro-1H-isoquinolin-2-yl)-carbamic acid 4-tert-butoxycarbonylamino-phenyl ester IC50: 3 nM 664316 3.1.1.79 0.000005 - (S)-4-isopropyl-3-methyl-2-[3-methylpiperidine-1-carbonyl]isoxazol-5[2H]-one - 703222 3.1.1.79 0.000005 - benzyl (4-[[(morpholin-4-ylamino)carbonyl]oxy]phenyl)acetate IC50: 5 nM 664316 3.1.1.79 0.000008 - 3-(4-chlorophenyl)-N,N-dimethyl-5-(methylsulfanyl)-1H-1,2,4-triazole-1-carboxamide - 703222 3.1.1.79 0.00001 - 4-[(cyclohexylcarbonyl)amino]phenyl morpholin-4-ylcarbamate IC50: 10 nM 664316 3.1.1.79 0.000019 - 4-chlorophenyl 3,4-dihydroisoquinolin-2(1H)-ylcarbamate IC50: 19 nM 664316 3.1.1.79 0.000024 - N',N'-bis-(2-butylamino-ethyl)-hydrazinecarboxylic acid 4-chloro-phenyl ester IC50: 24 nM 664316 3.1.1.79 0.000025 - trans-cyclipostin P pH 7.4, 37°C 750035