2.4.2.30 0.00018 - 4-amino-1,8-naphthalimide IC50: 0.00018 mM 637997 2.4.2.30 0.0003 - 2H-benz[c]isoquinolin-1-one IC50: 0.0003 mM 637997 2.4.2.30 0.0003 - 6(5H)-phenanthridinone IC50: 0.0003 mM 637997 2.4.2.30 0.00035 - 2-nitro-6(5H)-phenanthridione IC50: 0.00035 mM 637997 2.4.2.30 0.00039 - 1,5-dihydroxyisoquinoline IC50: 0.00039 mM 637997 2.4.2.30 0.0014 - 1,8-naphthalimide IC50: 0.0014 mM 637997 2.4.2.30 0.0014 - 2H-benz[de]isoquinoline-1,3-dione IC50: 0.0014 mM 637997 2.4.2.30 0.0019 - vitamin K1 IC50: 0.0019 mM 637997 2.4.2.30 0.007 - 1-hydroxyisoquinoline IC50: 0.007 mM 637997 2.4.2.30 0.0081 - 2,4(1H,3H)-quinazolinedione IC50: 0.0081 mM 637997 2.4.2.30 0.0081 - benzoyleneurea IC50: 0.0081 mM 637997 2.4.2.30 0.0085 - Chlorthenoxazin IC50: 0.0085 mM 637997 2.4.2.30 0.0091 - 3-Hydroxybenzamide IC50: 0.0091 mM 637997 2.4.2.30 0.0095 - 4-hydroxyquinazoline IC50: 0.0095 mM 637997 2.4.2.30 0.012 - 1(2H)-phthalazinone IC50: 0.012 mM 637997 2.4.2.30 0.012 - 3-Acetamidobenzamide IC50: 0.012 mM 637997 2.4.2.30 0.017 - 3-Methoxybenzamide IC50: 0.017 mM 637997 2.4.2.30 0.022 - 2-phenylchromone IC50: 0.022 mM 637997 2.4.2.30 0.022 - flavone IC50: 0.022 mM 637997 2.4.2.30 0.023 - 3-Aminophthalhydrazide IC50: 0.023 mM 637997 2.4.2.30 0.03 - 2,3-dihydro-1,4-phthalazinedione IC50: 0.03 mM 637997 2.4.2.30 0.043 - 5-iodouridine IC50: 0.043 mM 637997 2.4.2.30 0.044 - 2-mercapto-4(3H)-quinazolinone IC50: 0.044 mM 637997 2.4.2.30 0.045 - 2-methyl-1,4-benzopyrone IC50: 0.045 mM 637997 2.4.2.30 0.045 - 2-methylchromone IC50: 0.045 mM 637997 2.4.2.30 0.045 - 5-acetamidosalicylamide IC50: 0.045 mM 637997 2.4.2.30 0.048 - linoleic acid IC50: 0.048 mM 637997 2.4.2.30 0.05 - m-phthalamide IC50: 0.05 mM 637997 2.4.2.30 0.055 - 3-bromobenzamide IC50: 0.055 mM 637997 2.4.2.30 0.056 - 2-methyl-4(3H)-quinazolinone IC50: 0.056 mM 637997 2.4.2.30 0.071 - 5-Iodouracil IC50: 0.071 mM 637997 2.4.2.30 0.072 - 3-nitrophthalhydrazide IC50: 0.072 mM 637997 2.4.2.30 0.074 - 4-hydroxy-2-methylquinoline IC50: 0.074 mM 637997 2.4.2.30 0.08 - 4-hydroxyquinoline IC50: 0.08 mM 637997 2.4.2.30 0.082 - oleic acid IC50: 0.082 mM 637997 2.4.2.30 0.095 - palmitoleic acid IC50: 0.095 mM 637997 2.4.2.30 0.1 - 5-aminosalicylamide IC50: 0.1 mM 637997 2.4.2.30 0.11 - linolenic acid IC50: 0.11 mM 637997 2.4.2.30 0.12 - 2-fluorobenzamide IC50: 0.12 mM 637997 2.4.2.30 0.12 - 3-(N,N-dimethylamino)benzamide IC50: 0.12 mM 637997 2.4.2.30 0.12 - gamma-linolenic acid IC50: 0.12 mM 637997 2.4.2.30 0.15 - 2,3-benzodiazine IC50: 0.15 mM 637997 2.4.2.30 0.16 - 3-nitrobenzamide IC50: 0.16 mM 637997 2.4.2.30 0.16 - 5-Bromouracil IC50: 0.16 mM 637997 2.4.2.30 0.18 - 2,6-difluorobenzamide IC50: 0.18 mM 637997 2.4.2.30 0.18 - thymidine IC50: 0.18 mM 637997 2.4.2.30 0.19 - 3-Methylbenzamide IC50: 0.19 mM 637997 2.4.2.30 0.19 - 4,8-dihydroxy-2-quinolinecarboxylic acid IC50: 0.19 mM 637997 2.4.2.30 0.19 - 5-chlorosalicylamide IC50: 0.19 mM 637997 2.4.2.30 0.2 - 2-Methoxybenzamide IC50: 0.2 mM 637997 2.4.2.30 0.2 - 3-Fluorobenzamide IC50: 0.2 mM 637997 2.4.2.30 0.2 - 4-fluorobenzamide IC50: 0.2 mM 637997 2.4.2.30 0.21 - 5-Bromouridine IC50: 0.21 mM 637997 2.4.2.30 0.21 - nicotinamide IC50: 0.21 mM 637997 2.4.2.30 0.22 - 3-Chlorobenzamide IC50: 0.22 mM 637997 2.4.2.30 0.22 - Benzamide IC50: 0.22 mM 637997 2.4.2.30 0.25 - 1,4-naphthalenedione IC50: 0.25 mM 637997 2.4.2.30 0.25 - 5-hydroxy-1,4-naphthoquinone IC50: 0.25 mM 637997 2.4.2.30 0.25 - alpha-picolinamide IC50: 0.25 mM 637997 2.4.2.30 0.26 - 2,3-dichloro-1,4-naphthoquinone IC50: 0.26 mM 637997 2.4.2.30 0.27 - 5-Chlorouracil IC50: 0.27 mM 637997 2.4.2.30 0.28 - 4-hydroxybenzamide IC50: 0.28 mM 637997 2.4.2.30 0.29 - 4-aminophthalhydrazide IC50: 0.29 mM 637997 2.4.2.30 0.29 - 5-methyluracil IC50: 0.29 mM 637997 2.4.2.30 0.3 - 4-chlorobenzamide IC50: 0.3 mM 637997 2.4.2.30 0.31 - 3,4-dihydro-1(2H)-naphthalenone IC50: 0.31 mM 637997 2.4.2.30 0.33 - 2-Hydroxy-1,4-naphthoquinone IC50: 0.33 mM 637997 2.4.2.30 0.33 - 3-aminobenzamide IC50: 0.33 mM 637997 2.4.2.30 0.35 - 5-Methylnicotinamide IC50: 0.35 mM 637997 2.4.2.30 0.4 - 1,4-benzoquinone IC50: 0.4 mM 637997 2.4.2.30 0.42 - 2-methyl-1,4-naphthoquinone IC50: 0.42 mM 637997 2.4.2.30 0.42 - vitamin K3 IC50: 0.42 mM 637997 2.4.2.30 0.43 - 5-Nitrouracil IC50: 0.43 mM 637997 2.4.2.30 0.45 - all-trans-retinal IC50: 0.45 mM 637997 2.4.2.30 0.45 - N-hydroxynaphthalimide sodium salt IC50: 0.45 mM 637997 2.4.2.30 0.46 - carbonylsalicylamide IC50: 0.46 mM 637997 2.4.2.30 0.51 - 4-nitrophthalhydrazide IC50: 0.51 mM 637997 2.4.2.30 0.52 - 2-methyl-3-phytyl-1,4-naphthoquinone IC50: 0.52 mM 637997 2.4.2.30 0.56 - 3,5-dibromosalicylamide IC50: 0.56 mM 637997 2.4.2.30 0.56 - chromone-2-carboxylic acid IC50: 0.56 mM 637997 2.4.2.30 0.57 - 4-Hydroxycoumarin IC50: 0.57 mM 637997 2.4.2.30 0.6 - m-hydroxyacetophenone IC50: 0.6 mM 637997 2.4.2.30 0.62 - cyclohexanecarboxamide IC50: 0.62 mM 637997 2.4.2.30 0.62 - thiobenzamide IC50: 0.62 mM 637997 2.4.2.30 0.65 - 2-Aminobenzamide IC50: 0.65 mM 637997 2.4.2.30 0.67 - 4-hydroxy-2-quinolinecarboxylic acid IC50: 0.67 mM 637997 2.4.2.30 0.7 - 5-Hydroxy-2-methyl-1,4-naphthoquinone IC50: 0.7 mM 637997 2.4.2.30 0.72 - 4-chromanone IC50: 0.72 mM 637997 2.4.2.30 0.72 - menadione sodium bisulfite IC50: 0.72 mM 637997 2.4.2.30 0.79 - reserpine IC50: 0.79 mM 637997 2.4.2.30 0.81 - 1-Indanone IC50: 0.81 mM 637997 2.4.2.30 0.82 - 2-amino-3-chloro-1,4-naphthoquinone IC50: 0.82 mM 637997 2.4.2.30 0.82 - 2-hydroxybenzamide IC50: 0.82 mM 637997 2.4.2.30 0.85 - 6-aminocoumarin IC50: 0.85 mM 637997 2.4.2.30 0.93 - m-acetamidoacetophenone IC50: 0.93 mM 637997 2.4.2.30 0.99 - Isonicotinamide IC50: 0.99 mM 637997 2.4.2.30 1 - 2-acetamidobenzamide IC50: 1.0 mM 637997 2.4.2.30 1 - 2-chlorobenzamide IC50: 1.0 mM 637997 2.4.2.30 1 - phthalamide IC50: 1.0 mM 637997 2.4.2.30 1.1 - 4-methoxybenzamide IC50: 1.1 mM 637997 2.4.2.30 1.1 - 6-aminonicotinamide IC50: 1.1 mM 637997 2.4.2.30 1.2 - 3,5-dimethoxybenzamide IC50: 1.2 mM 637997 2.4.2.30 1.3 - 1,3-dihydroxynaphthalene IC50: 1.3 mM 637997 2.4.2.30 1.3 - 1-hydroxy-2-methyl-4-aminonaphthalene IC50: 1.3 mM 637997 2.4.2.30 1.4 - 8-acetamidocarsalam IC50: 1.4 mM 637997 2.4.2.30 1.5 - 2-methylbenzamide IC50: 1.5 mM 637997 2.4.2.30 1.6 - 3-nitrosalicylamide IC50: 1.6 mM 637997 2.4.2.30 1.8 - 4-Aminobenzamide IC50: 1.8 mM 637997 2.4.2.30 1.8 - 4-methylbenzamide IC50: 1.8 mM 637997 2.4.2.30 1.8 - N-(2-chloroethyl)1,8-naphthalamide IC50: above 1.8 mM 637997 2.4.2.30 1.8 - Thionicotinamide IC50: 1.8 mM 637997 2.4.2.30 1.9 - m-aminoacetophenone IC50: 1.9 mM 637997 2.4.2.30 2 - 1,3-benzodiazine IC50: 2.0 mM 637997 2.4.2.30 2 - 3-acetamidosalicylamide IC50: 2.0 mM 637997 2.4.2.30 2.2 - 2-trichloromethyl-4(3H)-quinazolinone IC50: 2.2 mM 637997 2.4.2.30 2.2 - 4-bromobenzamide IC50: 2.2 mM 637997 2.4.2.30 2.2 - novobiocin IC50: 2.2 mM, 5 mM, 90% inhibition in presence of Mg2+, 59% inhibition in absence of Mg2+ 637997 2.4.2.30 2.3 - 4-hydroxypyridine IC50: 2.3 mM 637997 2.4.2.30 2.3 - acetophenone IC50: 2.3 mM 637997 2.4.2.30 2.5 - 3,5-dinitrobenzamide IC50: 2.5 mM 637997 2.4.2.30 2.8 - 1,2-benzopyrone IC50: 2.8 mM 637997 2.4.2.30 2.9 - 2-bromobenzamide IC50: 2.9 mM 637997 2.4.2.30 3.8 - 1-methylnicotinamide chloride IC50: 3.8 mM 637997 2.4.2.30 4.3 - trans-decahydro-1-naphthalenone IC50: 4.3 mM 637997 2.4.2.30 4.7 - norharman IC50: 4.7 mM 637997 2.4.2.30 0.0033 - Benzamide IC50: 0.0033 mM 638001 2.4.2.30 0.0034 - 3-Methoxybenzamide IC50: 0.0034 mM 638001 2.4.2.30 0.0054 - 3-aminobenzamide IC50: 0.0054 638001 2.4.2.30 0.015 - 5-bromodeoxyuridine IC50: 0.015 mM 638001 2.4.2.30 0.031 - nicotinamide IC50: 0.031 mM 638001 2.4.2.30 0.043 - thymidine IC50: 0.043 mM 638001 2.4.2.30 0.046 - theophylline IC50: 0.046 mM 638001 2.4.2.30 0.07 - 5-Methylnicotinamide IC50: 0.07 mM 638001 2.4.2.30 0.077 - Zn2+ ZnCl2, IC50: 0.077 mM 638001 2.4.2.30 0.1 - 2-Aminobenzamide IC50: 0.1 mM 638001 2.4.2.30 0.11 - Theobromine IC50: 0.11 mM 638001 2.4.2.30 0.13 - Pyrazinamide IC50: 0.13 mM 638001 2.4.2.30 0.4 - 4-Aminobenzamide IC50: 0.4 mM 638001 2.4.2.30 1.4 - Caffeine IC50: 1.4 mM 638001 2.4.2.30 1.7 - 1-methylnicotinamide chloride IC50: 1.7 mM 638001 2.4.2.30 1.7 - hypoxanthine IC50: 1.7 mM 638001 2.4.2.30 3.1 - 3-isobutyl-1-methylxanthine IC50: 3.1 mM 638001 2.4.2.30 4.8 - Isonicotinate hydrazide IC50: 4.8 mM 638001 2.4.2.30 7.8 - 8-Methylnicotinamide IC50: 7.8 mM 638001 2.4.2.30 0.22 - 3-amino-1,4-dimethyl-5H-pyrido[4,3-b]indole i.e. Trp-P-1, 94% inhibition at 5 mM, IC50: 0.22 mM 675627 2.4.2.30 2.2 - 3-amino-1-methyl-5H-pyrido[4,3-b]indole i.e. Trp-P-2, 34% activation at 1 mM, 7% inhibition at 5 mM, IC50: 2.2 mM 675627 2.4.2.30 0.003 - diosmin pH 6.0, 30°C 694800 2.4.2.30 0.006 - 4296-1011 pH 6.0, 30°C 694800 2.4.2.30 0.021 - everninic acid pH 6.0, 30°C 694800 2.4.2.30 0.023 - E216-5303 pH 6.0, 30°C 694800 2.4.2.30 0.02 - suramin 25°C, pH not specified in the publication 722786 2.4.2.30 0.0858 - N-(acridin-9-yl)-4-nitrobenzamide 25°C, pH not specified in the publication 722786 2.4.2.30 0.086 - N-[2-oxo-4-(phenylamino)-3,8a-dihydro-2H-chromen-3-yl]acetamide 25°C, pH not specified in the publication 722786 2.4.2.30 0.157 - V8 protease 25°C, pH not specified in the publication 722786 2.4.2.30 0.000232 - TIQ-A isoform ARDT7, pH and temperature not specified in the publication 736061 2.4.2.30 0.000745 - phenantridinone isoform ARDT10, pH and temperature not specified in the publication 736061 2.4.2.30 0.000925 - olaparib isoform ARDT7, pH and temperature not specified in the publication 736061 2.4.2.30 0.00114 - phenantridinone isoform ARDT7, pH and temperature not specified in the publication 736061 2.4.2.30 0.00118 - EB-47 isoform ARDT10, pH and temperature not specified in the publication 736061 2.4.2.30 0.00204 - olaparib isoform ARDT10, pH and temperature not specified in the publication 736061 2.4.2.30 0.019 - 3-(4-oxo-3,5,6,7-tetrahydro-4H-cyclopenta[4,5]thieno[2,3-d]pyrimidin-2-yl)propanoic acid at pH 7.5 and 22°C 736518 2.4.2.30 0.0249 - 4-(4-oxo-3,4-dihydroquinazolin-2-yl)butanoic acid at pH 7.5 and 22°C 736518 2.4.2.30 0.0479 - 3-(4-oxo-3,4,5,6,7,8-hexahydro[1]benzothieno[2,3-d]pyrimidin-2-yl)propanoic acid at pH 7.5 and 22°C 736518 2.4.2.30 0.0524 - 2-(3-hydroxypropyl)-3,5,6,7-tetrahydro-4H-cyclopenta[4,5]thieno[2,3-d]pyrimidin-4-one at pH 7.5 and 22°C 736518 2.4.2.30 0.135 - 3-(4-oxo-3,4-dihydroquinazolin-2-yl)propanoic acid at pH 7.5 and 22°C 736518 2.4.2.30 0.169 - 2-(3-hydroxypropyl)-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4(3H)-one at pH 7.5 and 22°C 736518 2.4.2.30 0.294 - 3-(4-methoxy-6,7-dihydro-5H-cyclopenta[4,5]thieno[2,3-d]pyrimidin-2-yl)propanoic acid at pH 7.5 and 22°C 736518 2.4.2.30 0.0009 - 3-(4-oxo-3,4-dihydroquinazolin-2-yl)-N-[(1S)-1-phenylethyl]propanamide pH and temperature not specified in the publication 736615 2.4.2.30 0.001 - N-[(2S)-1-hydroxy-3-phenylpropan-2-yl]-3-(4-oxo-3,4-dihydroquinazolin-2-yl)propanamide pH and temperature not specified in the publication 736615 2.4.2.30 0.0013 - 3-(4-oxo-3,4-dihydroquinazolin-2-yl)-N-[(1S)-1-(pyridin-2-yl)ethyl]propanamide pH and temperature not specified in the publication 736615 2.4.2.30 0.0022 - 3-(4-oxo-3,4-dihydroquinazolin-2-yl)-N-[(1S)-1-phenylpropyl]propanamide pH and temperature not specified in the publication 736615 2.4.2.30 0.0022 - methyl (2S)-2-[[3-(4-oxo-3,4-dihydroquinazolin-2-yl)propanoyl]amino]-3-phenylpropanoate pH and temperature not specified in the publication 736615 2.4.2.30 0.0038 - (2S)-2-[[3-(4-oxo-3,4-dihydroquinazolin-2-yl)propanoyl]amino]-3-phenylpropanamide pH and temperature not specified in the publication 736615 2.4.2.30 0.0096 - N-[(2S)-1-hydroxybutan-2-yl]-3-(4-oxo-3,4-dihydroquinazolin-2-yl)propanamide pH and temperature not specified in the publication 736615 2.4.2.30 0.0111 - N-[(2S)-1-hydroxypropan-2-yl]-3-(4-oxo-3,4-dihydroquinazolin-2-yl)propanamide pH and temperature not specified in the publication 736615 2.4.2.30 0.0132 - N-[1-[4-(1H-imidazol-1-yl)phenyl]ethyl]-3-(4-oxo-3,4-dihydroquinazolin-2-yl)propanamide pH and temperature not specified in the publication 736615 2.4.2.30 0.0144 - 3-(4-oxo-3,4-dihydroquinazolin-2-yl)-N-[1-(4-sulfamoylphenyl)ethyl]propanamide pH and temperature not specified in the publication 736615 2.4.2.30 0.0152 - 3-(4-oxo-3,4-dihydroquinazolin-2-yl)-N-[(1R)-1-phenylethyl]propanamide pH and temperature not specified in the publication 736615 2.4.2.30 0.1 - 3-(4-oxo-3,4-dihydroquinazolin-2-yl)-N-[(1R)-1-(pyridin-2-yl)ethyl]propanamide IC50 above 0.1 mM, pH and temperature not specified in the publication 736615 2.4.2.30 0.1 - N-[(1R)-2,3-dihydro-1H-inden-1-yl]-3-(4-oxo-3,4-dihydroquinazolin-2-yl)propanamide IC50 above 0.1 mM, pH and temperature not specified in the publication 736615 2.4.2.30 0.1 - N-[(1S)-2,3-dihydro-1H-inden-1-yl]-3-(4-oxo-3,4-dihydroquinazolin-2-yl)propanamide IC50 above 0.1 mM, pH and temperature not specified in the publication 736615 2.4.2.30 0.003 - 4-nitro-7-[(1-oxo-1lambda(5)-pyridin-2-yl)sulfanyl]-2,1,3-benzoxadiazole at pH 7.5 and 25°C 758573 2.4.2.30 0.0068 - 4,5,7,9-tetrahydro-2H-purine-2,8(3H)-dithione at pH 7.5 and 25°C 758573 2.4.2.30 0.02 - (1E,4E)-1,5-di(pyridin-3-yl)penta-1,4-dien-3-one at pH 7.5 and 25°C 758573 2.4.2.30 0.000329 - 4-[4-(1-aminoethenyl)phenoxy]benzamide pH and temperature not specified in the publication 759013 2.4.2.30 0.00018 - 4-(4-carbamoylphenoxy)benzoic acid pH and temperature not specified in the publication 759148 2.4.2.30 0.00023 - 4-[(2-fluorophenyl)methoxy]benzamide pH and temperature not specified in the publication 759148 2.4.2.30 0.00033 - 4-[4-(1-aminoethenyl)phenoxy]benzamide pH and temperature not specified in the publication 759148 2.4.2.30 0.00071 - 4-(4-formylphenoxy)benzamide pH and temperature not specified in the publication 759148 2.4.2.30 0.00072 - 4-butoxybenzamide pH and temperature not specified in the publication 759148 2.4.2.30 0.0011 - 4-phenoxybenzamide pH and temperature not specified in the publication 759148 2.4.2.30 0.0013 - 4-(4-aminophenoxy)benzamide pH and temperature not specified in the publication 759148 2.4.2.30 0.0013 - 4-[(propan-2-yl)oxy]benzamide pH and temperature not specified in the publication 759148 2.4.2.30 0.00135 - 4-[(pyridin-2-yl)methoxy]benzamide pH and temperature not specified in the publication 759148 2.4.2.30 0.0014 - 4-(4-methoxyphenoxy)benzamide pH and temperature not specified in the publication 759148 2.4.2.30 0.0014 - 4-(benzyloxy)benzamide pH and temperature not specified in the publication 759148 2.4.2.30 0.0014 - 4-[(naphthalen-1-yl)methoxy]benzamide pH and temperature not specified in the publication 759148 2.4.2.30 0.0017 - 4-(2-fluorophenoxy)benzamide pH and temperature not specified in the publication 759148 2.4.2.30 0.0018 - 4-(4-hydroxyphenoxy)benzamide pH and temperature not specified in the publication 759148 2.4.2.30 0.0019 - 4-(2-phenoxyethoxy)benzamide pH and temperature not specified in the publication 759148 2.4.2.30 0.002 - 4-[[4-(aminocarbonyl)benzyl]oxy]benzamide pH and temperature not specified in the publication 759148 2.4.2.30 0.0022 - 4-[(3-bromophenyl)methoxy]benzamide pH and temperature not specified in the publication 759148 2.4.2.30 0.0028 - 4-methoxybenzamide pH and temperature not specified in the publication 759148 2.4.2.30 0.0033 - 4-[(3-fluorophenyl)methoxy]benzamide pH and temperature not specified in the publication 759148 2.4.2.30 0.0035 - 4-ethoxybenzamide pH and temperature not specified in the publication 759148 2.4.2.30 0.0038 - 4-[(2-bromophenyl)methoxy]benzamide pH and temperature not specified in the publication 759148 2.4.2.30 0.0045 - 4-[(3,5-dimethylphenyl)methoxy]benzamide pH and temperature not specified in the publication 759148 2.4.2.30 0.0073 - 4-carbamoylphenyl benzoate pH and temperature not specified in the publication 759148 2.4.2.30 0.0079 - 4-[(4-fluorophenyl)methoxy]benzamide pH and temperature not specified in the publication 759148 2.4.2.30 0.0093 - 4-[(4-methylphenyl)methoxy]benzamide pH and temperature not specified in the publication 759148